SCHEMBL8552282

SCHEMBL8552282

Cc1ccnc(N2CCN(C(=O)CCc3c(C)n4c5c(cccc35)CCC4)CC2)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.59
PARP1 P09874 1/20 0.52
HTR2A P28223 1/20 0.50
HTR2C P28335 1/20 0.50
TSHR P16473 4/20 0.44
KDM4E B2RXH2 4/20 0.44
SMN1; SMN2 Q16637 4/20 0.42
HSD17B10 Q99714 2/20 0.42
ALDH1A1 P00352 2/20 0.42
LMNA P02545 2/20 0.42
TP53 P04637 1/20 0.42
HTT P42858 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
MCL1 Q07820 2/20 0.41
BCL2L1 Q07817 1/20 0.41
CPT2 P23786 1/20 0.40
CPT1A P50416 1/20 0.40
CPT1B Q92523 1/20 0.40
ATM Q13315 1/20 0.40
POLB P06746 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8554233 0.89 ALOX5 (0.53) ALOX5PARP1HTR2AHTR2CTSHR
SCHEMBL8557565 0.84 ALOX5 (0.77) ALOX5HTR2AHTR2CHSD17B10ALDH1A1
Hydrochloric Acid SCHEMBL8555007 0.84 ALOX5 (0.75) ALOX5HTR2AHTR2CHSD17B10ALDH1A1
SCHEMBL8554623 0.84 ALOX5 (0.70) ALOX5HTR2AHTR2CHSD17B10ALDH1A1
Hydrochloric Acid SCHEMBL9304050 0.83 ALOX5 (0.69) ALOX5HTR2AHTR2CHSD17B10ALDH1A1
SCHEMBL8554776 0.82 ALOX5 (0.73) ALOX5HTR2AHTR2CHSD17B10ALDH1A1
Hydrochloric Acid SCHEMBL8555946 0.81 ALOX5 (0.71) ALOX5HTR2AHTR2CHSD17B10ALDH1A1
SCHEMBL9304984 0.81 ALOX5 (0.45) ALOX5PARP1TSHRKDM4ESMN1; SMN2
SCHEMBL8556392 0.79 ALOX5 (0.59) ALOX5PARP1HTR2AHTR2CTSHR
SCHEMBL8554000 0.78 ALOX5 (0.55) ALOX5PARP1TSHRKDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0529452-B1 1,7-Condensed 3-(piperazinoalkyl)indol derivatives, process and intermediates for their preparation and pharmaceutical compositions containing them SOLVAY PHARM GMBH (DE) 1998-11-11 EP disclosed
US-5324725-A Antiinflammatory agent, antiallergen KALI-CHEMIE PHARMA GMBH (DE) 1994-06-28 US disclosed
EP-0529452-A2 1,7-Condensed 2-(piperazinoalkyl)indol derivatives, process and intermediates for their preparation and pharmaceutical compositions containing them Kali-Chemie Pharma GmbH (DE) 1993-03-03 EP disclosed