SCHEMBL8552461

SCHEMBL8552461

O=C(OC1CCN(Cc2ccccc2)CC1)c1ccccc1Br

nearest known ligand 0.58

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
BCHE P06276 2/20 0.58
SCN1A P35498 2/20 0.53
SCN2A Q99250 2/20 0.53
SCN3A Q9NY46 2/20 0.53
SIGMAR1 Q99720 1/20 0.52
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
KDM4E B2RXH2 2/20 0.47
HSD17B10 Q99714 1/20 0.47
ALDH1A1 P00352 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8551440 0.99 BCHE (0.57) BCHESCN1ASCN2ASCN3ASIGMAR1
SCHEMBL8551865 0.86 BCHE (0.60) BCHESCN1ASCN2ASCN3ASIGMAR1
SCHEMBL8551876 0.85 BCHE (0.58) BCHESCN1ASCN2ASCN3ASIGMAR1
SCHEMBL8551180 0.85 BCHE (0.58) BCHESCN1ASCN2ASCN3ASIGMAR1
SCHEMBL8551916 0.85 SIGMAR1 (0.62) BCHESCN1ASCN2ASCN3ASIGMAR1
SCHEMBL8550391 0.85 POLB (0.62) BCHESCN1ASCN2ASCN3AKDM4E
Hydrochloric Acid SCHEMBL8551643 0.85 BCHE (0.58) BCHESCN1ASCN2ASCN3ASIGMAR1
Hydrochloric Acid SCHEMBL8550401 0.84 BCHE (0.57) BCHESCN1ASCN2ASCN3ASIGMAR1
Hydrochloric Acid SCHEMBL8552833 0.84 SIGMAR1 (0.61) BCHESCN1ASCN2ASCN3ASIGMAR1
Hydrochloric Acid SCHEMBL8556314 0.84 POLB (0.61) BCHESCN1ASCN2ASCN3AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753679-A SCIZOPHRENIA HOFFMANN-LA ROCHE INC. (US) 1998-05-19 US claimed
CN-1084329-C Benzyl piepridine derivs as pharmaceutical agents HOFFMANN LA ROCHE (CH) 2002-05-08 CN disclosed
EP-0871613-A1 BENZYL PIPERIDINE DERIVATIVES AS PHARMACEUTICAL AGENTS F. HOFFMANN-LA ROCHE AG (CH) 1998-10-21 EP disclosed
CN-1183768-A Benzyl piepridine derivs as pharmaceutical agents HOFFMANN LA ROCHE (CH) 1998-06-03 CN disclosed
US-5753679-A SCIZOPHRENIA HOFFMANN-LA ROCHE INC. (US) 1998-05-19 US disclosed
WO-1996035666-A1 BENZYL PIPERIDINE DERIVATIVES AS PHARMACEUTICAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 1996-11-14 WO disclosed