SCHEMBL8552660

SCHEMBL8552660

O=S(=O)(CCCOc1ccccc1)C(F)(F)F

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNA3 P22001 1/20 0.52
HDAC1 Q13547 3/20 0.49
HDAC2 Q92769 3/20 0.49
MGLL Q99685 1/20 0.46
PKM P14618 1/20 0.44
HDAC3 O15379 1/20 0.43
HDAC4 P56524 1/20 0.43
HDAC7 Q8WUI4 1/20 0.43
HDAC10 Q969S8 1/20 0.43
HDAC11 Q96DB2 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
HDAC9 Q9UKV0 1/20 0.43
HDAC5 Q9UQL6 1/20 0.43
DRD2 P14416 1/20 0.43
DRD4 P21917 1/20 0.43
DRD3 P35462 1/20 0.43
ALDH1A1 P00352 2/20 0.42
TAAR1 Q96RJ0 1/20 0.42
RECQL P46063 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8552394 0.91 KCNA3 (0.48) KCNA3HDAC1HDAC2MGLLPKM
SCHEMBL9080146 0.79 KCNA3 (0.52) KCNA3HDAC1HDAC2MGLLHDAC3
SCHEMBL7399184 0.78 TSHR (0.44) MGLL
SCHEMBL18889128 0.76 KCNA3 (0.48) KCNA3HDAC1HDAC2PKMALDH1A1
SCHEMBL7245161 0.76 KCNA3 (0.58) KCNA3HDAC1HDAC2PKMHDAC3
SCHEMBL7728981 0.76 KCNA3 (0.58) KCNA3HDAC1HDAC2MGLLPKM
SCHEMBL3085704 0.76 KCNA3 (0.58) KCNA3HDAC1HDAC2MGLLPKM
SCHEMBL20572659 0.76 KCNA3 (0.58) KCNA3HDAC1HDAC2MGLLPKM
SCHEMBL5704316 0.76 KCNA3 (0.58) KCNA3HDAC1HDAC2MGLLPKM
Potassium Ion SCHEMBL10575515 0.74 KCNA3 (0.56) KCNA3HDAC1HDAC2MGLLPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0840725-A1 AZETIDINONE DERIVATIVES FOR THE TREATMENT OF ATHEROSCLEROSIS SMITHKLINE BEECHAM PLC (GB) 1998-05-13 EP disclosed
WO-1997002242-A1 AZETIDINONE DERIVATIVES FOR THE TREATMENT OF ATHEROSCLEROSIS SMITHKLINE BEECHAM PLC (GB) 1997-01-23 WO disclosed