SCHEMBL8552893

SCHEMBL8552893

O=C(O)CCN1CCC(NC(=O)c2nnc(C3CCNCC3)s2)CC1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 7/20 0.43
ADRA1D P25100 1/20 0.37
ADRA1A P35348 1/20 0.37
ADRA1B P35368 1/20 0.37
KDM1A O60341 2/20 0.36
CARM1 Q86X55 1/20 0.36
PRMT6 Q96LA8 1/20 0.36
ALDH1A1 P00352 1/20 0.35
TSHR P16473 1/20 0.35
ITGB3 P05106 3/20 0.34
ITGA2B P08514 3/20 0.34
UTS2R Q9UKP6 1/20 0.34
HPGDS O60760 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8552049 0.89 SMYD3 (0.43) SMYD3ALDH1A1TSHRUTS2RHPGDS
Hydrochloric Acid SCHEMBL8592818 0.88 SMYD3 (0.41) SMYD3CARM1PRMT6UTS2R
SCHEMBL8550362 0.83 SMYD3 (0.40) SMYD3ALDH1A1TSHRITGB3ITGA2B
SCHEMBL8550368 0.83 SMYD3 (0.40) SMYD3ALDH1A1TSHRITGB3ITGA2B
Hydrochloric Acid SCHEMBL8551138 0.82 SMYD3 (0.40) SMYD3ALDH1A1TSHRITGB3ITGA2B
SCHEMBL8549842 0.81 SMYD3 (0.41) SMYD3ADRA1DADRA1AADRA1BKDM1A
Hydrochloric Acid SCHEMBL8551719 0.81 SMYD3 (0.42) SMYD3ALDH1A1UTS2R
SCHEMBL8555209 0.79 KDM4E (0.36) SMYD3TSHR
SCHEMBL8551904 0.77 ALDH1A1 (0.51) ALDH1A1TSHR
Hydrochloric Acid SCHEMBL8592586 0.77 SMYD3 (0.37) SMYD3ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0858457-A1 5-MEMBERED HETEROCYCLES, PHARMACEUTICAL AGENTS CONTAINING SAID COMPOUNDS AND THE USE THEREOF AND METHODS OF PRODUCING THEM Dr. Karl Thomae GmbH (DE) 1998-08-19 EP disclosed
WO-1997015567-A1 5-MEMBERED HETEROCYCLES, PHARMACEUTICAL AGENTS CONTAINING SAID COMPOUNDS AND THE USE THEREOF AND METHODS OF PRODUCING THEM DR. KARL THOMAE GMBH (DE) 1997-05-01 WO disclosed