SCHEMBL8552049

SCHEMBL8552049

O=C(O)CN1CCC(NC(=O)c2nnc(C3CCNCC3)s2)CC1

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 9/20 0.43
CHRM5 P08912 1/20 0.36
CHRM3 P20309 1/20 0.36
SIGMAR1 Q99720 1/20 0.36
UTS2R Q9UKP6 5/20 0.35
HPGDS O60760 1/20 0.34
ALDH1A1 P00352 1/20 0.34
TSHR P16473 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8552893 0.89 SMYD3 (0.43) SMYD3UTS2RHPGDSALDH1A1TSHR
Hydrochloric Acid SCHEMBL8551719 0.87 SMYD3 (0.42) SMYD3CHRM5CHRM3SIGMAR1UTS2R
SCHEMBL8553958 0.85 GSK3B (0.42)
Hydrochloric Acid SCHEMBL8592818 0.81 SMYD3 (0.41) SMYD3UTS2R
SCHEMBL8550368 0.80 SMYD3 (0.40) SMYD3ALDH1A1TSHR
SCHEMBL8550362 0.80 SMYD3 (0.40) SMYD3ALDH1A1TSHR
Hydrochloric Acid SCHEMBL8551138 0.79 SMYD3 (0.40) SMYD3ALDH1A1TSHR
SCHEMBL8553962 0.78 ITGB3 (0.34) SIGMAR1
Hydrochloric Acid SCHEMBL8592586 0.78 SMYD3 (0.37) SMYD3ALDH1A1TSHR
SCHEMBL8555209 0.76 KDM4E (0.36) SMYD3TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0858457-A1 5-MEMBERED HETEROCYCLES, PHARMACEUTICAL AGENTS CONTAINING SAID COMPOUNDS AND THE USE THEREOF AND METHODS OF PRODUCING THEM Dr. Karl Thomae GmbH (DE) 1998-08-19 EP disclosed
WO-1997015567-A1 5-MEMBERED HETEROCYCLES, PHARMACEUTICAL AGENTS CONTAINING SAID COMPOUNDS AND THE USE THEREOF AND METHODS OF PRODUCING THEM DR. KARL THOMAE GMBH (DE) 1997-05-01 WO disclosed