SCHEMBL8553277

SCHEMBL8553277

CCCCN1CCC(c2csc3ccc(NC(=O)c4ccccc4Br)cc23)CC1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.49
SLC6A4 P31645 1/20 0.49
F2R P25116 5/20 0.45
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
TSHR P16473 1/20 0.41
HTR1D P28221 7/20 0.41
KMT2A Q03164 1/20 0.41
ALDH1A1 P00352 3/20 0.41
HTR1B P28222 5/20 0.41
CHRM2 P08172 1/20 0.41
NPY2R P49146 1/20 0.40
HPGD P15428 2/20 0.39
KDM4E B2RXH2 1/20 0.39
USP2 O75604 1/20 0.39
TP53 P04637 1/20 0.39
MAPK1 P28482 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8548023 0.89 DRD2 (0.50) DRD2SLC6A4HTR1DKMT2AHTR1B
SCHEMBL8552547 0.87 DRD2 (0.47) DRD2SLC6A4HTR1DKMT2AHTR1B
SCHEMBL8548076 0.86 DRD2 (0.47) DRD2SLC6A4HTR1DHTR1BCHRM2
SCHEMBL8703019 0.85 DRD2 (0.53) DRD2SLC6A4NPC1RAB9AKDM4E
SCHEMBL8547861 0.83 DRD2 (0.50) DRD2SLC6A4F2R
SCHEMBL7479962 0.83 HTR1D (0.62) DRD2HTR1DHTR1BCHRM2
SCHEMBL8702974 0.82 DRD2 (0.53) DRD2SLC6A4NPC1RAB9AHTR1D
SCHEMBL8708757 0.81 DRD2 (0.53) DRD2SLC6A4ALDH1A1
SCHEMBL8552559 0.80 DRD2 (0.47) DRD2SLC6A4HTR1DALDH1A1HTR1B
SCHEMBL8553349 0.80 DRD2 (0.47) DRD2SLC6A4NPC1SMN1; SMN2HTR1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5792763-A MIGRAINES; ANALGESICS; DISEASES LINKED TO DECREASED NEUROTRANMISSION OF SEROTONIN IN MAMMALS ELI LILLY AND COMPANY (US) 1998-08-11 US disclosed
WO-1998015545-A1 NEW SEROTONIN 5-HT1F AGONISTS ELI LILLY AND COMPANY (US) 1998-04-16 WO disclosed
EP-0835869-A2 New serotonin 5-HT1F agonists ELI LILLY AND COMPANY (US) 1998-04-15 EP disclosed