SCHEMBL8553492

SCHEMBL8553492

COc1ccc(-c2c(C(=O)O)n(Cc3ccc4nsnc4c3)c3cccc(O)c23)cc1

nearest known ligand 0.64

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
EDNRB P24530 10/20 0.64
EDNRA P25101 7/20 0.54
PTGES O14684 1/20 0.39
PPARG P37231 3/20 0.39
TP53 P04637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8551194 0.91 EDNRB (0.64) EDNRBEDNRAPTGESTP53
SCHEMBL8553494 0.88 EDNRB (0.52) EDNRBEDNRAPPARGTP53
SCHEMBL8553006 0.87 EDNRB (0.62) EDNRBEDNRA
SCHEMBL8549014 0.87 EDNRB (0.61) EDNRBEDNRAPPARG
SCHEMBL8547579 0.86 EDNRB (0.64) EDNRBEDNRA
SCHEMBL8550885 0.84 EDNRB (0.74) EDNRBEDNRATP53
SCHEMBL6313759 0.83 EDNRB (0.62) EDNRBEDNRAPTGESPPARGTP53
SCHEMBL8550228 0.83 EDNRB (0.85) EDNRBEDNRA
SCHEMBL8548527 0.83 EDNRB (0.73) EDNRBEDNRATP53
SCHEMBL6316183 0.83 EDNRB (0.61) EDNRBEDNRAPPARGTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863898-A1 ENDOTHELIN RECEPTOR ANTAGONISTS MERCK PATENT GmbH (DE) 1998-09-16 EP disclosed
WO-1997019077-A1 ENDOTHELIN RECEPTOR ANTAGONISTS MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1997-05-29 WO disclosed