SCHEMBL8554024

SCHEMBL8554024

Fc1ccc(-c2nnc(Cl)c3cc(Cl)c(Cl)cc23)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 5/20 0.41
ADORA1 P30542 5/20 0.41
ADORA2B P29275 2/20 0.41
ADORA3 P0DMS8 2/20 0.41
ALDH1A1 P00352 2/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
GABRA1 P14867 1/20 0.38
TACR2 P21452 1/20 0.38
OPRD1 P41143 1/20 0.38
KMT5B Q4FZB7 1/20 0.38
KMT5C Q86Y97 1/20 0.38
SMN1; SMN2 Q16637 4/20 0.37
NPC1 O15118 4/20 0.37
RAB9A P51151 4/20 0.37
TP53 P04637 2/20 0.37
TSHR P16473 1/20 0.37
HSD17B10 Q99714 1/20 0.37
THRB P10828 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4837981 0.86 ADORA2A (0.41) ADORA2AADORA1ADORA2BADORA3ALDH1A1
SCHEMBL8551380 0.81 LMNA (0.45) ADORA2AADORA1ADORA2BADORA3ALDH1A1
SCHEMBL1268020 0.80 ESR1 (0.49) ADORA2AALDH1A1MEN1KMT2ANPSR1
SCHEMBL4840257 0.77 MAPK14 (0.46) ADORA2AADORA1ADORA2BADORA3ALDH1A1
SCHEMBL8548298 0.77 PLAU (0.40) ADORA2AADORA1ADORA2BADORA3ALDH1A1
SCHEMBL7914983 0.75 NPSR1 (0.53) ALDH1A1MEN1KMT2ANPSR1SMN1; SMN2
SCHEMBL8548292 0.74 ADORA2A (0.41) ADORA2AADORA1ADORA2BADORA3ALDH1A1
SCHEMBL9139946 0.73 SMN1; SMN2 (0.41) ADORA2AADORA1ADORA2BADORA3ALDH1A1
SCHEMBL30170698 0.73 AHR (0.41) ALDH1A1MEN1KMT2ATP53TSHR
SCHEMBL6591372 0.73 AHR (0.41) ALDH1A1MEN1KMT2ATP53TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825187-A1 Condensed pyridazinyl guanidines, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-25 EP disclosed