SCHEMBL8554724

SCHEMBL8554724

COC(=O)CCc1nc2c(=O)[nH]c3cc(C(F)(F)F)ccc3n2c1C

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 2/20 0.48
PDE9A O76083 2/20 0.48
KDM4E B2RXH2 3/20 0.43
ALDH1A1 P00352 2/20 0.43
HSD17B10 Q99714 2/20 0.43
HPGD P15428 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
EGFR P00533 2/20 0.43
CHEK1 O14757 1/20 0.37
DAPK3 O43293 1/20 0.37
PRKD3 O94806 1/20 0.37
MET P08581 1/20 0.37
PDGFRA P16234 1/20 0.37
FLT1 P17948 1/20 0.37
LTK P29376 1/20 0.37
GRK5 P34947 1/20 0.37
CDK8 P49336 1/20 0.37
PRKX P51817 1/20 0.37
NEK2 P51955 1/20 0.37
LIMK1 P53667 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8554829 0.89 PDE9A (0.61) PDE5APDE9AMEN1CYP1A2HSP90AA1
SCHEMBL8557784 0.86 PDE5A (0.47) PDE5APDE9AALDH1A1MEN1CYP1A2
SCHEMBL8555426 0.80 CHEK1 (0.49) KDM4EALDH1A1HSD17B10HPGDSMN1; SMN2
SCHEMBL7505355 0.79 PDE5A (0.52) PDE5APDE9AALDH1A1CHEK1DAPK3
SCHEMBL31328139 0.79 PDE5A (0.52) PDE5APDE9AALDH1A1CHEK1DAPK3
SCHEMBL8558570 0.79 KDM4E (0.48) PDE5APDE9AKDM4EALDH1A1HSD17B10
SCHEMBL7503779 0.79 CHEK1 (0.55) PDE5APDE9ACHEK1DAPK3PRKD3
SCHEMBL7517883 0.79 PDE5A (0.48) PDE5APDE9AALDH1A1CHEK1DAPK3
SCHEMBL8557418 0.77 PDE5A (0.49) PDE5APDE9AALDH1A1HPGDMEN1
SCHEMBL8556953 0.76 PDE5A (0.48) PDE5APDE9AALDH1A1CHEK1DAPK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0691970-B1 IMIDAZOLOQUINOXALINONE DERIVATIVES AS EAA ANTAGONISTS BASF AG (DE) 1998-11-11 EP disclosed