SCHEMBL8558570

SCHEMBL8558570

CCOC(=O)CCc1nc2c(=O)[nH]c3cc(C(F)(F)F)ccc3n2c1-c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.48
HSD17B10 Q99714 4/20 0.48
LMNA P02545 2/20 0.48
ALDH1A1 P00352 2/20 0.48
PDE5A O76074 2/20 0.46
PDE9A O76083 2/20 0.46
GRIN1 Q05586 2/20 0.40
GRIN2B Q13224 2/20 0.40
MAPT P10636 1/20 0.40
HPGD P15428 2/20 0.40
S1PR4 O95977 1/20 0.40
TP53 P04637 1/20 0.40
S1PR1 P21453 1/20 0.40
MAPK1 P28482 1/20 0.40
STAT3 P40763 1/20 0.40
STAT1 P42224 1/20 0.40
KMT2A Q03164 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
TLR9 Q9NR96 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8553493 0.89 PDE9A (0.58) KDM4EALDH1A1PDE5APDE9AHPGD
SCHEMBL8554950 0.84 PDE5A (0.44) KDM4EHSD17B10ALDH1A1PDE5APDE9A
SCHEMBL8557199 0.83 PDE5A (0.43) KDM4EALDH1A1PDE5APDE9AGRIN1
SCHEMBL9080716 0.80 PDE9A (0.54) KDM4EHSD17B10LMNAALDH1A1PDE5A
SCHEMBL8554724 0.79 PDE5A (0.48) KDM4EHSD17B10LMNAALDH1A1PDE5A
SCHEMBL8554829 0.78 PDE9A (0.61) PDE5APDE9AMAPTKMT2ANPSR1
SCHEMBL8555764 0.78 PDE5A (0.49) KDM4EALDH1A1PDE5APDE9AMAPT
SCHEMBL8557792 0.77 PDE5A (0.47) KDM4EALDH1A1PDE5APDE9AMAPT
SCHEMBL3588054 0.77 PDE9A (0.52) KDM4EHSD17B10LMNAALDH1A1PDE5A
SCHEMBL7503779 0.76 CHEK1 (0.55) PDE5APDE9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0691970-B1 IMIDAZOLOQUINOXALINONE DERIVATIVES AS EAA ANTAGONISTS BASF AG (DE) 1998-11-11 EP disclosed