SCHEMBL8555004

SCHEMBL8555004

CC(C)(C)OC(=O)N1CCN(CC(=O)Nc2c(Cl)cc(N)cc2Cl)CC1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.57
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49
KDM4E B2RXH2 4/20 0.48
MAPT P10636 2/20 0.48
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
CHRM2 P08172 1/20 0.45
CHRM4 P08173 1/20 0.45
CHRM1 P11229 1/20 0.45
CHRM3 P20309 1/20 0.45
HSD17B10 Q99714 2/20 0.43
MAPK1 P28482 2/20 0.43
USP2 O75604 1/20 0.43
LMNA P02545 1/20 0.43
HPGD P15428 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
CETP P11597 1/20 0.42
POLB P06746 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8553179 0.85 ALDH1A1 (0.53) ALDH1A1NPC1RAB9AKDM4EMAPT
SCHEMBL29106576 0.78 RAD52 (0.67) ALDH1A1KDM4EMEN1KMT2ACHRM2
SCHEMBL18072532 0.78 CHRM3 (0.53) ALDH1A1KDM4EMAPTMEN1KMT2A
SCHEMBL15986885 0.77 F13A1 (0.49) ALDH1A1NPC1RAB9AMAPTCHRM2
SCHEMBL211276 0.76 KCNT1 (0.56) ALDH1A1NPC1RAB9AKDM4EMAPT
SCHEMBL8556919 0.76 NPC1 (0.56) ALDH1A1NPC1RAB9AKDM4EMAPT
SCHEMBL6846616 0.75 MEN1 (0.47) ALDH1A1MAPTMEN1KMT2AUSP2
SCHEMBL16577075 0.75 MEN1 (0.62) ALDH1A1NPC1RAB9AKDM4EMAPT
SCHEMBL15629359 0.75 CHRM2 (0.50) ALDH1A1NPC1RAB9AKDM4EMAPT
SCHEMBL209299 0.74 KDM4E (0.61) ALDH1A1KDM4EKMT2ACHRM2CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0582164-B1 Adenosine re-uptake inhibiting derivatives of diphenyl oxazoles, thiazoles and imidazoles BRISTOL MYERS SQUIBB CO (US) 1998-12-23 EP disclosed
EP-0582164-A1 Adenosine re-uptake inhibiting derivatives of diphenyl oxazoles, thiazoles and imidazoles Bristol-Myers Squibb Company (US) 1994-02-09 EP disclosed