SCHEMBL8553179

SCHEMBL8553179

CC(C)(C)OC(=O)N1CCN(CC(=O)Nc2c(Cl)cc([N+](=O)[O-])cc2Cl)CC1

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.53
MAPT P10636 6/20 0.49
LMNA P02545 4/20 0.49
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
KDM4E B2RXH2 2/20 0.45
GAA P10253 3/20 0.44
GFER P55789 1/20 0.43
MCL1 Q07820 1/20 0.43
GLA P06280 1/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
CHRM2 P08172 1/20 0.42
CHRM4 P08173 1/20 0.42
CHRM1 P11229 1/20 0.42
CHRM3 P20309 1/20 0.42
HTT P42858 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8555004 0.85 ALDH1A1 (0.57) ALDH1A1MAPTLMNANPC1RAB9A
SCHEMBL9255657 0.83 SLC29A1 (0.41) ALDH1A1MAPTLMNAMEN1KMT2A
SCHEMBL29106529 0.80 ALDH1A1 (0.56) ALDH1A1MAPTLMNAGAAGLA
SCHEMBL8558093 0.78 NPC1 (0.51) ALDH1A1MAPTLMNANPC1RAB9A
SCHEMBL12005556 0.78 ALDH1A1 (0.64) ALDH1A1MAPTLMNAMEN1KMT2A
SCHEMBL7801883 0.78 NPC1 (0.53) ALDH1A1MAPTLMNANPC1RAB9A
Hydrochloric Acid SCHEMBL7519848 0.77 NPC1 (0.52) ALDH1A1MAPTLMNANPC1RAB9A
SCHEMBL13861942 0.74 ALDH1A1 (0.58) ALDH1A1MAPTLMNAKDM4EMEN1
SCHEMBL31639389 0.74 ALDH1A1 (0.70) ALDH1A1MAPTLMNAGAAMEN1
SCHEMBL18072532 0.74 CHRM3 (0.53) ALDH1A1MAPTLMNAKDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0582164-B1 Adenosine re-uptake inhibiting derivatives of diphenyl oxazoles, thiazoles and imidazoles BRISTOL MYERS SQUIBB CO (US) 1998-12-23 EP disclosed
EP-0582164-A1 Adenosine re-uptake inhibiting derivatives of diphenyl oxazoles, thiazoles and imidazoles Bristol-Myers Squibb Company (US) 1994-02-09 EP disclosed