SCHEMBL8555957

SCHEMBL8555957

COc1cc2ncnc(Nc3ccc4nn(Cc5ccccc5)nc4c3)c2cc1OC

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 6/20 0.71
EGFR P00533 11/20 0.63
KDR P35968 7/20 0.63
RET P07949 2/20 0.63
LCK P06239 2/20 0.61
EPHA2 P29317 3/20 0.61
EPHB4 P54760 3/20 0.61
CLK1 P49759 2/20 0.60
ABCG2 Q9UNQ0 1/20 0.60
RIPK2 O43353 1/20 0.59
EPHB2 P29323 1/20 0.59
FBP1 P09467 2/20 0.58
AURKA O14965 1/20 0.58
INSR P06213 1/20 0.58
PDGFRB P09619 1/20 0.58
FLT4 P35916 1/20 0.58
TEK Q02763 1/20 0.58
AURKB Q96GD4 1/20 0.58
KIF5B P33176 1/20 0.58
GAK O14976 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8557888 0.83 ERBB2 (1.00) ERBB2EGFRKDRRETLCK
SCHEMBL8096166 0.83 EGFR (0.62) ERBB2EGFR
SCHEMBL8933754 0.81 EGFR (0.80) ERBB2EGFRKDRRETLCK
SCHEMBL8556365 0.81 ERBB2 (0.69) ERBB2EGFRKDRRETLCK
SCHEMBL8560764 0.81 ERBB2 (0.72) ERBB2EGFRKDRRETLCK
SCHEMBL1387156 0.81 EGFR (0.75) ERBB2EGFRKDRRETLCK
SCHEMBL8309598 0.80 EGFR (0.65) ERBB2EGFRKDRRETLCK
Hydrochloric Acid SCHEMBL8810665 0.80 EGFR (0.79) ERBB2EGFRKDRRETLCK
SCHEMBL18158179 0.80 EGFR (0.79) ERBB2EGFRKDRRETLCK
Hydrochloric Acid SCHEMBL8811182 0.80 EGFR (0.76) ERBB2EGFRKDRRETLCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0843671-A1 HETEROCYCLIC COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GLAXO GROUP LIMITED (GB) 1998-05-27 EP claimed
WO-1997003069-A1 HETEROCYCLIC COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GLAXO GROUP LIMITED (GB) 1997-01-30 WO claimed
EP-0843671-A1 HETEROCYCLIC COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GLAXO GROUP LIMITED (GB) 1998-05-27 EP disclosed
WO-1997003069-A1 HETEROCYCLIC COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GLAXO GROUP LIMITED (GB) 1997-01-30 WO disclosed