SCHEMBL8560764

SCHEMBL8560764

COc1cc2ncnc(Nc3ccc4c(c3)nnn4Cc3ccccc3)c2cc1OC

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 6/20 0.72
EGFR P00533 12/20 0.59
KDR P35968 4/20 0.59
RET P07949 1/20 0.59
LCK P06239 3/20 0.58
CLK1 P49759 1/20 0.56
ABCG2 Q9UNQ0 1/20 0.56
EPHA2 P29317 1/20 0.56
EPHB4 P54760 1/20 0.56
LMNA P02545 3/20 0.56
MAPT P10636 3/20 0.56
MAPK1 P28482 3/20 0.56
ALDH1A1 P00352 2/20 0.56
HTT P42858 2/20 0.56
POLB P06746 1/20 0.56
ERBB4 Q15303 1/20 0.56
RIPK2 O43353 1/20 0.56
EPHB2 P29323 1/20 0.56
FLT1 P17948 1/20 0.54
KDM4E B2RXH2 3/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8556365 0.92 ERBB2 (0.69) ERBB2EGFRKDRRETLCK
SCHEMBL8555349 0.84 ERBB2 (1.00) ERBB2EGFRKDRRETLMNA
SCHEMBL8093486 0.83 EGFR (0.57) ERBB2EGFRLMNAMAPTMAPK1
Hydrochloric Acid SCHEMBL31681715 0.83 ERBB2 (0.98) ERBB2EGFRKDRRETLCK
SCHEMBL8555957 0.81 ERBB2 (0.71) ERBB2EGFRKDRRETLCK
SCHEMBL8556847 0.81 ERBB2 (1.00) ERBB2EGFRKDRRETLCK
Hydrochloric Acid SCHEMBL8596174 0.80 ERBB2 (0.98) ERBB2EGFRKDRRETLCK
SCHEMBL8595567 0.79 ERBB2 (0.86) ERBB2EGFRKDRRETLCK
SCHEMBL1387156 0.78 EGFR (0.75) ERBB2EGFRKDRRETLCK
Hydrochloric Acid SCHEMBL8558936 0.78 ERBB2 (0.84) ERBB2EGFRKDRRETLCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0843671-A1 HETEROCYCLIC COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GLAXO GROUP LIMITED (GB) 1998-05-27 EP claimed
WO-1997003069-A1 HETEROCYCLIC COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GLAXO GROUP LIMITED (GB) 1997-01-30 WO claimed
EP-0843671-A1 HETEROCYCLIC COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GLAXO GROUP LIMITED (GB) 1998-05-27 EP disclosed
WO-1997003069-A1 HETEROCYCLIC COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GLAXO GROUP LIMITED (GB) 1997-01-30 WO disclosed