SCHEMBL8555980

SCHEMBL8555980

O=C(OC1CCN(Cc2ccc(Br)cc2)CC1)c1ccc(F)cc1

nearest known ligand 0.70

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.56
HTR2A P28223 1/20 0.53
GAA P10253 1/20 0.49
SIGMAR1 Q99720 2/20 0.49
SLC6A12 P48065 1/20 0.49
TMEM97 Q5BJF2 1/20 0.49
MCHR1 Q99705 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8550562 0.99 ADRB2 (0.55) ADRB2HTR2AGAASIGMAR1SLC6A12
SCHEMBL8549980 0.90 GPR183 (0.60) SIGMAR1
SCHEMBL8553837 0.89 SCN1A (0.60) ADRB2GAA
Hydrochloric Acid SCHEMBL8550815 0.89 GPR183 (0.58) SIGMAR1
SCHEMBL8550198 0.89 ADRB2 (0.57) ADRB2HTR2AGAA
SCHEMBL8549828 0.89 CHRM2 (0.59) SIGMAR1
SCHEMBL8551089 0.89 CARM1 (0.57) SIGMAR1
Hydrochloric Acid SCHEMBL8553600 0.88 SCN1A (0.59) ADRB2GAA
Hydrochloric Acid SCHEMBL8551048 0.88 ADRB2 (0.56) ADRB2HTR2AGAA
Hydrochloric Acid SCHEMBL8554706 0.88 KMT2A (0.58) SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1084329-C Benzyl piepridine derivs as pharmaceutical agents HOFFMANN LA ROCHE (CH) 2002-05-08 CN disclosed
EP-0871613-A1 BENZYL PIPERIDINE DERIVATIVES AS PHARMACEUTICAL AGENTS F. HOFFMANN-LA ROCHE AG (CH) 1998-10-21 EP disclosed
CN-1183768-A Benzyl piepridine derivs as pharmaceutical agents HOFFMANN LA ROCHE (CH) 1998-06-03 CN disclosed
US-5753679-A SCIZOPHRENIA HOFFMANN-LA ROCHE INC. (US) 1998-05-19 US disclosed
WO-1996035666-A1 BENZYL PIPERIDINE DERIVATIVES AS PHARMACEUTICAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 1996-11-14 WO disclosed