SCHEMBL8553837

SCHEMBL8553837

Cc1ccc(C(=O)OC2CCN(Cc3ccc(Br)cc3)CC2)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN1A P35498 1/20 0.60
SCN2A Q99250 1/20 0.60
SCN3A Q9NY46 1/20 0.60
KDM4E B2RXH2 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.49
LMNA P02545 1/20 0.49
GPR183 P32249 2/20 0.49
ALDH1A1 P00352 2/20 0.48
MAPT P10636 1/20 0.48
PTPRF P10586 1/20 0.47
PTPN2 P17706 1/20 0.47
PTPN1 P18031 1/20 0.47
GAA P10253 1/20 0.47
MEN1 O00255 1/20 0.47
ADRB2 P07550 1/20 0.47
KMT2A Q03164 1/20 0.47
CARM1 Q86X55 1/20 0.46
PRMT6 Q96LA8 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
DRD4 P21917 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8553600 0.99 SCN1A (0.59) SCN1ASCN2ASCN3AKDM4ESMN1; SMN2
SCHEMBL8551183 0.94 SCN1A (0.68) SCN1ASCN2ASCN3AKDM4ESMN1; SMN2
Hydrochloric Acid SCHEMBL8553929 0.92 SCN1A (0.66) SCN1ASCN2ASCN3AKDM4ESMN1; SMN2
SCHEMBL8551160 0.89 SCN1A (0.61) SCN1ASCN2ASCN3AKDM4EGAA
SCHEMBL8555980 0.89 ADRB2 (0.56) GAAADRB2
SCHEMBL8553670 0.89 SCN1A (0.61) SCN1ASCN2ASCN3AKDM4ESMN1; SMN2
SCHEMBL8549980 0.89 GPR183 (0.60) LMNAGPR183PTPRFPTPN2PTPN1
Hydrochloric Acid SCHEMBL8550562 0.88 ADRB2 (0.55) GAAADRB2
Hydrochloric Acid SCHEMBL8550815 0.88 GPR183 (0.58) LMNAGPR183PTPRFPTPN2PTPN1
Hydrochloric Acid SCHEMBL8554961 0.88 SCN1A (0.60) SCN1ASCN2ASCN3AKDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1084329-C Benzyl piepridine derivs as pharmaceutical agents HOFFMANN LA ROCHE (CH) 2002-05-08 CN disclosed
EP-0871613-A1 BENZYL PIPERIDINE DERIVATIVES AS PHARMACEUTICAL AGENTS F. HOFFMANN-LA ROCHE AG (CH) 1998-10-21 EP disclosed
CN-1183768-A Benzyl piepridine derivs as pharmaceutical agents HOFFMANN LA ROCHE (CH) 1998-06-03 CN disclosed
US-5753679-A SCIZOPHRENIA HOFFMANN-LA ROCHE INC. (US) 1998-05-19 US disclosed
WO-1996035666-A1 BENZYL PIPERIDINE DERIVATIVES AS PHARMACEUTICAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 1996-11-14 WO disclosed