SCHEMBL8556224

SCHEMBL8556224

N#CC1(N)Cc2cccc3cccc(c23)C1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.39
TSHR P16473 2/20 0.39
BACE1 P56817 1/20 0.33
ALDH1A1 P00352 5/20 0.32
HPGD P15428 4/20 0.32
KDM4E B2RXH2 4/20 0.32
HSD17B10 Q99714 3/20 0.32
CYP1A2 P05177 2/20 0.32
CYP1A1 P04798 1/20 0.32
CYP1B1 Q16678 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
TYMS P04818 1/20 0.31
CYP2C19 P33261 1/20 0.31
GAA P10253 1/20 0.31
MAPT P10636 1/20 0.31
KMT2A Q03164 1/20 0.30
LMNA P02545 1/20 0.30
PARP1 P09874 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3308997 0.81 ALDH1A1 (0.38) TSHRALDH1A1HPGDGAAMAPT
SCHEMBL28896828 0.72 TSHR (0.41) CYP3A4TSHRALDH1A1HPGDKDM4E
SCHEMBL8558686 0.71 CYP3A4 (0.40) CYP3A4TSHRALDH1A1HPGDKDM4E
SCHEMBL8553587 0.69 BACE1 (0.39) TSHRBACE1ALDH1A1HPGDKMT2A
SCHEMBL15848208 0.69 CYP3A4 (0.35) CYP3A4TSHRBACE1ALDH1A1HPGD
SCHEMBL27538147 0.69 TSHR (0.46) CYP3A4TSHRALDH1A1HPGDKDM4E
SCHEMBL27577152 0.69 TSHR (0.46) CYP3A4TSHRALDH1A1HPGDKDM4E
SCHEMBL27497708 0.68 TSHR (0.41) CYP3A4TSHRALDH1A1HPGDKDM4E
Hydrochloric Acid SCHEMBL9179624 0.68 BACE1 (0.38) TSHRBACE1ALDH1A1HPGDKMT2A
Acenaphthene SCHEMBL27875520 0.67 TSHR (0.55) CYP3A4TSHRALDH1A1HPGDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0635497-B1 Benzospiroalkene derivatives, process for their preparation and pharmaceutical compostions containing them ADIR (FR) 1998-05-20 EP disclosed
US-5436261-A Adrenergic agonists ADIR ET COMPAGNIE (FR) 1995-07-25 US disclosed
EP-0635497-A2 Benzospiroalkene derivatives, process for their preparation and pharmaceutical compostions containing them ADIR ET COMPAGNIE (FR) 1995-01-25 EP disclosed