SCHEMBL8553587

SCHEMBL8553587

N#CC1(N)CCc2ccccc2C1

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 4/20 0.39
ADRA2A P08913 2/20 0.38
SIGMAR1 Q99720 1/20 0.35
TSHR P16473 1/20 0.34
KDM1A O60341 2/20 0.34
MAOB P27338 1/20 0.34
ALDH1A1 P00352 3/20 0.34
HPGD P15428 1/20 0.34
KMT2A Q03164 1/20 0.33
PARP1 P09874 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9179624 0.98 BACE1 (0.38) BACE1ADRA2ASIGMAR1TSHRKDM1A
SCHEMBL3308997 0.86 ALDH1A1 (0.38) TSHRMAOBALDH1A1HPGDKMT2A
SCHEMBL16605583 0.79 KDM1A (0.41) BACE1KDM1A
SCHEMBL16605572 0.79 BACE1 (0.42) BACE1KDM1A
SCHEMBL8556494 0.78 KDM1A (0.41) BACE1KDM1A
SCHEMBL7918142 0.78 BACE1 (0.33) BACE1
SCHEMBL25762670 0.76 NAMPT (0.32)
SCHEMBL8653266 0.76 ADRA2A (0.50) ADRA2AKDM1A
SCHEMBL8620656 0.74 ADRA2A (0.48) ADRA2A
SCHEMBL8650675 0.74 LMNA (0.36) TSHRALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0635497-B1 Benzospiroalkene derivatives, process for their preparation and pharmaceutical compostions containing them ADIR (FR) 1998-05-20 EP disclosed
EP-0635497-A2 Benzospiroalkene derivatives, process for their preparation and pharmaceutical compostions containing them ADIR ET COMPAGNIE (FR) 1995-01-25 EP disclosed
EP-0435988-A1 2-AMINO-7-CARBAMOYL-1,2,3,4-TETRAHYDRONAPHTHALENES, PROCESS FOR PREPARING THEM AND THEIR USE AS DRUGS BOEHRINGER INGELHEIM KG (DE) 1991-07-10 EP disclosed
WO-1991001297-A1 2-AMINO-7-CARBAMOYL-1,2,3,4-TETRAHYDRONAPHTHALENES, PROCESS FOR PREPARING THEM AND THEIR USE AS DRUGS BOEHRINGER INGELHEIM KG (DE) 1991-02-07 WO disclosed