SCHEMBL8556535

SCHEMBL8556535

O=C(Nc1ccc(C(=O)N2CCc3cncnc3-c3ccccc32)cc1)c1ccccc1Cl

nearest known ligand 0.60

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 6/20 0.52
AVPR1B P47901 1/20 0.52
AVPR2 P30518 5/20 0.51
OXTR P30559 2/20 0.49
HSD11B1 P28845 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8562567 0.92 AVPR2 (0.48) AVPR1AAVPR2OXTR
SCHEMBL8556396 0.91 AVPR2 (0.55) AVPR1AAVPR2
SCHEMBL8559368 0.89 AVPR1A (0.59) AVPR1AAVPR2OXTR
SCHEMBL8556714 0.85 ROCK2 (0.43) AVPR1AAVPR2
SCHEMBL8562670 0.84 AVPR1A (0.60) AVPR1AAVPR1BAVPR2OXTR
SCHEMBL8820731 0.83 AVPR1A (0.63) AVPR1AAVPR1BAVPR2OXTR
SCHEMBL8820363 0.77 AVPR2 (0.60) AVPR1AAVPR1BAVPR2OXTR
SCHEMBL8820823 0.77 AVPR2 (0.55) AVPR1AAVPR2
SCHEMBL7340204 0.76 AVPR1A (0.55) AVPR1AAVPR1BAVPR2
SCHEMBL8559859 0.76 AVPR2 (0.55) AVPR1AAVPR2OXTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640592-B1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID CO (US) 1998-12-30 EP disclosed
WO-1997047625-A1 TRICYCLIC BENZAZEPINE VASOPRESSIN ANTAGONISTS AMERICAN CYANAMID COMPANY (US) 1997-12-18 WO disclosed