SCHEMBL8556761

SCHEMBL8556761

Nc1cc2c(cc1Cl)NC(=O)C(=O)[N]2

nearest known ligand 0.38

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CES1 P23141 2/20 0.38
GAA P10253 1/20 0.37
CA12 O43570 1/20 0.30
CA9 Q16790 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8122389 0.85 CES1 (0.47) CES1
SCHEMBL8557868 0.79 CES1 (0.34) CES1
SCHEMBL8557286 0.76 CES1 (0.37) CES1
SCHEMBL8559761 0.74 AKR1B1 (0.40) CES1CA12CA9
SCHEMBL8128202 0.73 GRIN2D (0.41) CES1
SCHEMBL8554501 0.72 HTR2C (0.37) CES1
SCHEMBL8120664 0.72 EGFR (0.40)
SCHEMBL8556891 0.71 RET (0.37) CES1GAACA12CA9
SCHEMBL8123432 0.71 CES1 (0.37) CES1
SCHEMBL8127567 0.71 CES1 (0.37) CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0647137-A4 GLYCINE RECEPTOR ANTAGONISTS AND THE USE THEREOF. UNIV CALIFORNIA WEBER ECKARD (US) 1998-09-16 EP disclosed
EP-0647137-A1 GLYCINE RECEPTOR ANTAGONISTS AND THE USE THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1995-04-12 EP disclosed