SCHEMBL8557286

SCHEMBL8557286

O=C1[N]c2cc(Cl)c(F)cc2NC1=O

nearest known ligand 0.37

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CES1 P23141 2/20 0.37
ALPL P05186 1/20 0.32
MAPT P10636 1/20 0.32
ALDH1A1 P00352 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
TDP2 O95551 1/20 0.31
PGR P06401 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8122389 0.85 CES1 (0.47) CES1MAPTALDH1A1
SCHEMBL8121964 0.85
SCHEMBL8554501 0.79 HTR2C (0.37) CES1ALDH1A1
SCHEMBL8128202 0.77 GRIN2D (0.41) CES1
SCHEMBL6013572 0.76 PDE3B (0.33) CES1
SCHEMBL8556761 0.76 CES1 (0.38) CES1
SCHEMBL8118374 0.74 ESPL1 (0.38) MAPTALDH1A1TDP1PGR
SCHEMBL8120664 0.72 EGFR (0.40)
SCHEMBL8555842 0.71 KMT2A (0.39) CES1MAPT
SCHEMBL8124019 0.71 GRIN2D (0.30) CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0647137-A4 GLYCINE RECEPTOR ANTAGONISTS AND THE USE THEREOF. UNIV CALIFORNIA WEBER ECKARD (US) 1998-09-16 EP disclosed
EP-0647137-A1 GLYCINE RECEPTOR ANTAGONISTS AND THE USE THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1995-04-12 EP disclosed