SCHEMBL8557868

SCHEMBL8557868

Nc1cc2c(cc1Br)NC(=O)C(=O)[N]2

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 2/20 0.34
BCHE P06276 1/20 0.34
TGM2 P21980 1/20 0.33
MEN1 O00255 1/20 0.32
APAF1 O14727 1/20 0.32
ALDH1A1 P00352 1/20 0.32
POLB P06746 1/20 0.32
MAPT P10636 1/20 0.32
THRB P10828 1/20 0.32
NR4A1 P22736 1/20 0.32
RECQL P46063 1/20 0.32
BLM P54132 1/20 0.32
KMT2A Q03164 1/20 0.32
PTPN11 Q06124 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
CASP7 P55210 1/20 0.31
CASP6 P55212 1/20 0.31
CASP8 Q14790 1/20 0.31
TYMS P04818 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8554584 0.85 CES1 (0.38) CES1BCHETGM2
SCHEMBL8556761 0.79 CES1 (0.38) CES1
SCHEMBL8555748 0.74 ALDH1A1 (0.40) CES1BCHEMEN1ALDH1A1MAPT
SCHEMBL8556891 0.71 RET (0.37) CES1TGM2MEN1ALDH1A1MAPT
SCHEMBL8121964 0.71
SCHEMBL8122389 0.71 CES1 (0.47) CES1TGM2MEN1ALDH1A1MAPT
SCHEMBL8128045 0.71 POLB (0.38) CES1BCHEPOLB
SCHEMBL5528413 0.69 CES1 (0.62) CES1BCHETGM2ALDH1A1POLB
SCHEMBL8121209 0.68 GRIN2D (0.35) MEN1ALDH1A1POLBMAPTKMT2A
SCHEMBL8557274 0.68 ALDH1A1 (0.30) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0647137-A4 GLYCINE RECEPTOR ANTAGONISTS AND THE USE THEREOF. UNIV CALIFORNIA WEBER ECKARD (US) 1998-09-16 EP disclosed
EP-0647137-A1 GLYCINE RECEPTOR ANTAGONISTS AND THE USE THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1995-04-12 EP disclosed