SCHEMBL8556980

SCHEMBL8556980

CCn1c2nc(-c3cccnc3)[nH]c2c(=O)n2nc(Cc3ccccc3)nc12

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 12/20 0.51
ADORA1 P30542 8/20 0.51
ALDH1A1 P00352 3/20 0.51
TSHR P16473 2/20 0.51
KDM4E B2RXH2 2/20 0.51
CYP1A2 P05177 2/20 0.51
CYP3A4 P08684 2/20 0.51
HSD17B10 Q99714 2/20 0.51
HPGD P15428 1/20 0.51
MAPK1 P28482 1/20 0.51
THPO P40225 1/20 0.51
PMP22 Q01453 1/20 0.51
ADORA2A P29274 9/20 0.46
MEN1 O00255 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
KMT2A Q03164 1/20 0.45
ADORA3 P0DMS8 4/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7668670 0.93 ADORA2B (0.51) ADORA2BADORA1ALDH1A1TSHRKDM4E
SCHEMBL8559651 0.91 ADORA2B (0.61) ADORA2BADORA1ALDH1A1TSHRKDM4E
SCHEMBL8561695 0.89 ADORA2B (0.54) ADORA2BADORA1ALDH1A1TSHRKDM4E
SCHEMBL7670431 0.82 ADORA2B (0.54) ADORA2BADORA1ALDH1A1TSHRKDM4E
SCHEMBL8562832 0.78 ADORA2B (0.43) ADORA2BADORA1ALDH1A1TSHRKDM4E
SCHEMBL7659412 0.75 ADORA2B (0.45) ADORA2BADORA1ALDH1A1TSHRKDM4E
SCHEMBL7671642 0.74 ADORA2A (0.42) ADORA2BADORA1ADORA2AADORA3
SCHEMBL7665201 0.71 ADORA2A (0.45) ADORA2BADORA2AKMT2AADORA3
SCHEMBL7662113 0.70 ADORA1 (0.51) ADORA2BADORA1TSHRCYP1A2PMP22
SCHEMBL1321894 0.69 ADORA2B (1.00) ADORA2BADORA1ALDH1A1TSHRKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0880524-A1 NEW TRIAZOLOPURINES, METHOD OF PREPARING THEM AND THEIR USE AS DRUGS Boehringer Ingelheim Pharma KG (DE) 1998-12-02 EP disclosed
WO-1998003511-A1 NEW TRIAZOLOPURINES, METHOD OF PREPARING THEM AND THEIR USE AS DRUGS BOEHRINGER INGELHEIM PHARMA KG (DE) 1998-01-29 WO disclosed