SCHEMBL8557958

SCHEMBL8557958

Cc1ncc(CCCOc2c(C)cc(-c3nnn(C)n3)cc2C)o1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
NPC1 O15118 1/20 0.32
NFKB1 P19838 1/20 0.32
RAB9A P51151 1/20 0.32
NFKB2 Q00653 1/20 0.32
RELA Q04206 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
EPHX2 P34913 1/20 0.31
FFAR1 O14842 1/20 0.31
GRIN1 Q05586 1/20 0.30
GRIN2B Q13224 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8824428 0.84 NR1I2 (0.39) NR1I2CYP3A4CYP2D6NPC1NFKB1
SCHEMBL8824438 0.83 NR1I2 (0.39) NR1I2CYP3A4CYP2D6NPC1NFKB1
SCHEMBL8824414 0.83 NR1I2 (0.39) NR1I2CYP3A4CYP2D6NPC1NFKB1
SCHEMBL8552034 0.82 NR1I2 (0.35) NR1I2CYP3A4CYP2D6NPC1NFKB1
SCHEMBL9089893 0.82 NR1I2 (0.59) NR1I2CYP3A4CYP2D6NPC1NFKB1
SCHEMBL8603712 0.82 NR1I2 (0.37) NR1I2CYP3A4CYP2D6NPC1NFKB1
SCHEMBL9078729 0.81 RAB9A (0.41) NR1I2CYP3A4CYP2D6NPC1NFKB1
SCHEMBL9089930 0.80 NR1I2 (0.35) NR1I2CYP3A4CYP2D6NPC1NFKB1
SCHEMBL8558294 0.79 NR1I2 (0.41) NR1I2CYP3A4CYP2D6NPC1NFKB1
SCHEMBL14191677 0.78 NR1I2 (0.45) NR1I2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5846986-A Therapeutic phenoxyalkylazoles and phenoxyalkylazines SANOFI (FR) 1998-12-08 US disclosed
US-5721261-A TREATING PICORNAVIRUS INFECTIONS SANOFI PHARMACEUTICALS, INC. (US) 1998-02-24 US disclosed
US-5552420-A TREATING PICORNAVIRAL INFECTIONS STERLING WINTHROP INC. (US) 1996-09-03 US disclosed
WO-1995031452-A1 THERAPEUTIC PHENOXYALKYLAZOLES AND PHENOXYALKYLAZINES SANOFI WINTHROP, INC. (US) 1995-11-23 WO disclosed