SCHEMBL8558249

SCHEMBL8558249

Cc1ccc(C(=O)N(C)c2ccc(C(=O)N3Cc4ccccc4Cc4ccccc43)cc2)c(C)c1

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.45
HPGD P15428 1/20 0.45
RAB9A P51151 1/20 0.45
KMT2A Q03164 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
AVPR1A P37288 7/20 0.43
AVPR2 P30518 5/20 0.43
HSP90AA1 P07900 1/20 0.43
PDK1 Q15118 1/20 0.43
KCNN4 O15554 1/20 0.40
KCNA3 P22001 1/20 0.40
BCL2 P10415 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8557534 0.91 AVPR2 (0.45) NPC1HPGDRAB9AKMT2ASMN1; SMN2
SCHEMBL8561629 0.91 AVPR2 (0.52) NPC1HPGDRAB9AKMT2ASMN1; SMN2
SCHEMBL8561048 0.90 AVPR2 (0.48) AVPR1AAVPR2HSP90AA1PDK1
SCHEMBL8561249 0.86 AVPR2 (0.50) AVPR1AAVPR2
SCHEMBL8562797 0.84 AVPR2 (0.54) AVPR1AAVPR2HSP90AA1PDK1
SCHEMBL8557707 0.84 ALDH1A1 (0.47) RAB9ASMN1; SMN2AVPR1AAVPR2
SCHEMBL8563827 0.84 ALDH1A1 (0.47) NPC1HPGDRAB9AKMT2ASMN1; SMN2
SCHEMBL7333788 0.84 AVPR1A (0.66) AVPR1AAVPR2
SCHEMBL8559548 0.83 POLB (0.51) HPGDAVPR1AAVPR2HSP90AA1PDK1
SCHEMBL8561685 0.83 AVPR1A (0.44) NPC1HPGDRAB9AKMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640592-B1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID CO (US) 1998-12-30 EP disclosed