SCHEMBL8558357

SCHEMBL8558357

COC(=O)CC1(C2CCCCC2=O)CNC(=O)N1c1ccc2c(c1)CCN(C(=O)C(F)(F)F)CC2

nearest known ligand 0.37

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 3/20 0.37
ESR2 Q92731 3/20 0.37
PDE4B Q07343 1/20 0.32
PDE4D Q08499 1/20 0.32
NR3C2 P08235 1/20 0.31
HSD11B1 P28845 1/20 0.30
HDAC6 Q9UBN7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8563245 0.83 ESR1 (0.38) ESR1ESR2PDE4BPDE4DNR3C2
SCHEMBL8567149 0.72 ESR1 (0.38) ESR1ESR2PDE4BPDE4DHSD11B1
SCHEMBL8559776 0.71 HTR6 (0.35) HDAC6
SCHEMBL8565993 0.71 ESR1 (0.40) ESR1ESR2HDAC6
Hydrochloric Acid SCHEMBL8564477 0.71 HTR6 (0.34) HDAC6
Hydrochloric Acid SCHEMBL8569203 0.70 HTR6 (0.34)
Hydrochloric Acid SCHEMBL8564921 0.69 INSR (0.34)
SCHEMBL8559199 0.69 ESR1 (0.39) ESR1ESR2PDE4BPDE4D
SCHEMBL8561377 0.68 ESR1 (0.41) ESR1ESR2HDAC6
SCHEMBL8563251 0.68 ESR1 (0.39) ESR1ESR2PDE4BPDE4DHDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5827849-A HAVING INHIBITORY EFFECT ON INFLAMMATION AND BONE DEGRADATION, ANTITHROMBOTIC, ANTIAGGREGATORY AND TUMOR- OR METASTASIS-INHIBITING EFFECT KARL THOMAE GMBH (DE) 1998-10-27 US disclosed