SCHEMBL8558465

SCHEMBL8558465

Nc1ccc(Sc2cccc3ccccc23)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.51
HPGD P15428 2/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
DHFR P00374 4/20 0.49
CYP3A4 P08684 2/20 0.48
TSHR P16473 2/20 0.48
MAPK1 P28482 2/20 0.48
SIRT2 Q8IXJ6 1/20 0.47
SIRT1 Q96EB6 1/20 0.47
SIRT3 Q9NTG7 1/20 0.47
IFNAR1 P17181 1/20 0.44
ALDH1A1 P00352 2/20 0.43
KEAP1 Q14145 1/20 0.43
HSD17B10 Q99714 1/20 0.43
PDE7A Q13946 1/20 0.43
LMNA P02545 1/20 0.42
NPY1R P25929 1/20 0.42
NPY2R P49146 1/20 0.42
HTR6 P50406 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2890325 0.84 IFNAR1 (0.49) HPGDDHFRCYP3A4TSHRMAPK1
SCHEMBL31490493 0.84 IFNAR1 (0.49) HPGDDHFRCYP3A4TSHRMAPK1
SCHEMBL9814281 0.81 CYP3A4 (0.65) KDM1AHPGDCYP2C9CYP2C19DHFR
SCHEMBL28393840 0.81 IFNAR1 (0.44) KDM1AHPGDTSHRMAPK1SIRT2
SCHEMBL7201257 0.81 NR1H2 (0.48) CYP2C9CYP2C19DHFRMAPK1SIRT2
SCHEMBL13730600 0.81 SMN1; SMN2 (0.47) CYP2C9CYP2C19DHFRCYP3A4MAPK1
SCHEMBL9923541 0.81 IFNAR1 (0.47) CYP2C9DHFRCYP3A4MAPK1SIRT2
SCHEMBL28850516 0.81 DHFR (0.46) HPGDDHFRCYP3A4TSHRMAPK1
SCHEMBL9814267 0.79 CYP3A4 (0.70) KDM1AHPGDCYP2C9CYP2C19DHFR
SCHEMBL31167972 0.79 IFNAR1 (0.60) HPGDCYP2C9CYP2C19CYP3A4TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5814646-A TREATING THE PROGRESSION OF ALZHEIMER'S DISEASE, BRAIN DISORDERS ELI LILLY AND COMPANY (US) 1998-09-29 US disclosed
US-5624937-A TREATMENT OF ALZHEIMER'S DISEASE ELI LILLY AND COMPANY (US) 1997-04-29 US disclosed
EP-0013414-B1 UREA DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR USE AS INSECTICIDES CELAMERCK GmbH & Co. KG (DE) 1982-06-23 EP disclosed
US-4275077-A Insecticidal acyl urea derivatives CELAMERCK GMBH & CO. KG (DE) 1981-06-23 US disclosed
EP-0013414-A2 Urea derivatives, process for their preparation and their use as insecticides CELAMERCK GmbH & Co. KG (DE) 1980-07-23 EP disclosed