SCHEMBL8558472

SCHEMBL8558472

O=S(=O)(Cl)c1nc2ncccn2n1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
PDE10A Q9Y233 2/20 0.39
ALDH1A1 P00352 2/20 0.39
TSHR P16473 1/20 0.39
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
HPGD P15428 2/20 0.37
KDM4E B2RXH2 1/20 0.36
APOBEC3A P31941 1/20 0.36
APOBEC3G Q9HC16 1/20 0.36
LMNA P02545 1/20 0.34
USP2 O75604 1/20 0.34
SMN1; SMN2 Q16637 3/20 0.33
MAPT P10636 1/20 0.32
HTR6 P50406 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5225420 0.83 NPC1 (0.40) NPC1RAB9APDE10AALDH1A1TSHR
SCHEMBL6552357 0.79 HPGD (0.40) NPC1RAB9APDE10AALDH1A1TSHR
SCHEMBL10519274 0.75 ALDH1A1 (0.40) NPC1RAB9APDE10AALDH1A1TSHR
SCHEMBL8355273 0.74 SMN1; SMN2 (0.41) ALDH1A1MEN1KMT2AHPGDKDM4E
SCHEMBL3190914 0.74 ALDH1A1 (0.47) NPC1RAB9AALDH1A1MEN1KMT2A
SCHEMBL8881888 0.73 KDM4E (0.46) ALDH1A1TSHRMEN1KMT2AHPGD
SCHEMBL7840633 0.71 JAK2 (0.45) NPC1RAB9APDE10AALDH1A1MEN1
SCHEMBL10660778 0.71 HPGD (0.40) NPC1RAB9AALDH1A1HPGDKDM4E
SCHEMBL8113305 0.71 HTR6 (0.36) ALDH1A1LMNAUSP2HTR6
SCHEMBL8559896 0.71 MAP4K4 (0.33) NPC1RAB9AMEN1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 34 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0630377-A1 TRIAZOLOPYRIMIDINESULFONAMIDES AS HERBICIDES CIBA-GEIGY AG (CH) 1994-12-28 EP claimed
WO-1993016079-A1 TRIAZOLOPYRIMIDINESULFONAMIDES AS HERBICIDES CIBA-GEIGY AG (CH) 1993-08-19 WO claimed
EP-0142811-A2 Method of preparing 1,2,4-triazolo [1,5-a] - pyrimidine-2-sulfonyl chlorides THE DOW CHEMICAL COMPANY (US) 1985-05-29 EP claimed
JP-60172984-A None JP disclosed
EP-0537611-B1 Process for the preparation of substituted N-(aryl)-1,2,4-triazolopyrimidine-2-sulfonamides DOW AGROSCIENCES LLC (US) 1998-08-12 EP disclosed
US-5602075-A N-aryl[1,2,4]triazolo[1,5-a]pyrazine-2-sulfonamide herbicides DOWELANCO (US) 1997-02-11 US disclosed
EP-0630377-A1 TRIAZOLOPYRIMIDINESULFONAMIDES AS HERBICIDES CIBA-GEIGY AG (CH) 1994-12-28 EP disclosed
EP-0340828-B1 5-Fluoromethyl-1,2,4-triazolo(1,5-a)-pyrimidine-2-sulfonamides, process for their preparation and compositions for their use as herbicides DOWELANCO (US) 1994-03-02 EP disclosed
WO-1993016079-A1 TRIAZOLOPYRIMIDINESULFONAMIDES AS HERBICIDES CIBA-GEIGY AG (CH) 1993-08-19 WO disclosed
EP-0537611-A1 Process for the preparation of substituted N-(aryl)-1,2,4-triazolopyrimidine-2-sulfonamides DOWELANCO (US) 1993-04-21 EP disclosed
US-5177206-A Process for the preparation of substituted N-(aryl)-1,2,4-triazolopyrimidine-2-sulfonamides DOWELANCO (US) 1993-01-05 US disclosed
US-4740233-A Substituted 1,2,4-triazolo[1,5-a]-pyrimidine-2-sulfonamides and compositions and methods of controlling undesired vegetation and suppressing the nitrification of ammonium nitrogen in soil THE DOW CHEMICAL COMPANY (US) 1988-04-26 US disclosed
US-4734123-A HERBICIDE THE DOW CHEMICAL COMPANY (US) 1988-03-29 US disclosed
EP-0142811-A3 Method of preparing 1,2,4-triazolo [1,5-a] - pyrimidine-2-sulfonyl chlorides THE DOW CHEMICAL COMPANY (US) 1986-03-12 EP disclosed
EP-0142811-A3 Method of preparing 1,2,4-triazolo [1,5-a] - pyrimidine-2-sulfonyl chlorides THE DOW CHEMICAL COMPANY (US) 1986-03-12 EP disclosed
JP-S60172984-A MANUFACTURE OF 1,2,4-TRIAZOLO(1,5-A)- PYRIMIDINE-2-SULFONYLCHLORIDE DOW CHEMICAL CO 1985-09-06 JP disclosed
EP-0142811-A2 Method of preparing 1,2,4-triazolo [1,5-a] - pyrimidine-2-sulfonyl chlorides THE DOW CHEMICAL COMPANY (US) 1985-05-29 EP disclosed
EP-0142811-A2 Method of preparing 1,2,4-triazolo [1,5-a] - pyrimidine-2-sulfonyl chlorides THE DOW CHEMICAL COMPANY (US) 1985-05-29 EP disclosed
EP-0142811-A2 Method of preparing 1,2,4-triazolo [1,5-a] - pyrimidine-2-sulfonyl chlorides THE DOW CHEMICAL COMPANY (US) 1985-05-29 EP disclosed
EP-0142152-A2 Novel substituted 1,2,4-triazolo- [1,5-a] pyrimidine-2-sulfonamides and compositions and methods of controlling undesired vegetation and suppressing the nitrification of ammonium nitrogen in soil THE DOW CHEMICAL COMPANY (US) 1985-05-22 EP disclosed