SCHEMBL8558499

SCHEMBL8558499

COC(=O)Cc1ccccc1CC(=O)NCCc1cc(O)c(OC)c(OC)c1

nearest known ligand 0.57

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.57
LMNA P02545 3/20 0.52
ALDH1A1 P00352 2/20 0.52
HSD17B10 Q99714 1/20 0.52
KMT2A Q03164 5/20 0.51
MEN1 O00255 4/20 0.51
POLB P06746 4/20 0.49
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
HTT P42858 1/20 0.47
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C19 P33261 1/20 0.46
PTPN1 P18031 1/20 0.46
TDP1 Q9NUW8 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8558635 0.91 TAAR1 (0.70) TAAR1LMNAALDH1A1HSD17B10KMT2A
SCHEMBL10535357 0.84 CYP1A2 (0.64) TAAR1LMNAALDH1A1KMT2AMEN1
SCHEMBL8559166 0.83 LMNA (0.67) LMNAALDH1A1KMT2AMEN1CA1
SCHEMBL8556958 0.82 MEN1 (0.58) TAAR1LMNAALDH1A1HSD17B10KMT2A
SCHEMBL8558009 0.81 CA1 (0.69) LMNAKMT2AMEN1POLBCA1
SCHEMBL8556404 0.81 MEN1 (0.69) LMNAALDH1A1KMT2AMEN1CA1
SCHEMBL8553751 0.80 CA1 (0.65) LMNAALDH1A1KMT2AMEN1POLB
SCHEMBL8558286 0.80 LMNA (0.59) LMNAKMT2AMEN1CA1CA2
SCHEMBL10536452 0.79 TAAR1 (0.72) TAAR1ALDH1A1HSD17B10KMT2AMEN1
SCHEMBL8558637 0.79 LMNA (0.58) LMNAALDH1A1KMT2AMEN1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0617022-B1 6,7, dialkoxy-3,4-dihydroisoquinolin-8-ol, process for preparation thereof and process for preparation of 6,7-dialkoxy-1,2,3,4-tetrahydroisoquinolin-8-ol using the compound BANYU PHARMA CO LTD (JP) 1998-02-11 EP disclosed
US-5446164-A Regioselective cyclization of phenethylamide derivative in presence of phosphoric acid halide, reducing formed compound BANYU PHARMACEUTICAL CO., LTD. (JP) 1995-08-29 US disclosed
EP-0617022-A1 6,7, dialkoxy-3,4-dihydroisoquinolin-8-ol, process for preparation thereof and process for preparation of 6,7-dialkoxy-1,2,3,4-tetrahydroisoquinolin-8-ol using the compound BANYU PHARMACEUTICAL CO., LTD. (JP) 1994-09-28 EP disclosed