SCHEMBL8558930

SCHEMBL8558930

Cc1ccc(C(=O)Nc2ccc(C(=O)N3CCc4ccccc4-c4ccccc43)cc2)c(C)c1

nearest known ligand 0.83

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 2/20 0.60
OXTR P30559 2/20 0.60
AVPR1A P37288 2/20 0.60
NPC1 O15118 1/20 0.55
HPGD P15428 1/20 0.55
RAB9A P51151 1/20 0.55
KMT2A Q03164 1/20 0.55
SMN1; SMN2 Q16637 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8556628 0.91 AVPR2 (0.53) AVPR2OXTRAVPR1ANPC1HPGD
SCHEMBL8556989 0.91 AVPR1A (0.72) AVPR2OXTRAVPR1A
SCHEMBL8559258 0.90 AVPR2 (0.58) AVPR2OXTRAVPR1A
SCHEMBL8685905 0.90 AVPR2 (0.57) AVPR2OXTRAVPR1A
SCHEMBL8557460 0.87 AVPR1A (0.64) AVPR2OXTRAVPR1A
SCHEMBL8559570 0.85 AVPR1A (0.55) AVPR2OXTRAVPR1ANPC1HPGD
SCHEMBL8559975 0.85 AVPR2 (0.58) AVPR2OXTRAVPR1ANPC1HPGD
SCHEMBL8558289 0.84 AVPR2 (0.60) AVPR2OXTRAVPR1ARAB9A
SCHEMBL8563752 0.84 ALDH1A1 (0.57) AVPR2OXTRAVPR1A
SCHEMBL8557290 0.83 AVPR2 (0.64) AVPR2AVPR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640592-B1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID CO (US) 1998-12-30 EP disclosed
EP-0640592-A1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID COMPANY (US) 1995-03-01 EP disclosed