SCHEMBL8559006

SCHEMBL8559006

COc1cc(C(=O)N2Cc3ccccc3Cc3ccccc32)ccc1NC(=O)c1ccc(Cl)cc1Cl

nearest known ligand 0.75

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 9/20 0.75
AVPR1A P37288 8/20 0.75
PYGL P06737 2/20 0.51
KDM4E B2RXH2 1/20 0.49
ACHE P22303 1/20 0.49
HDAC1 Q13547 1/20 0.48
HDAC8 Q9BY41 1/20 0.48
HDAC6 Q9UBN7 1/20 0.48
SPTLC2 O15270 1/20 0.46
ALDH1A1 P00352 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8315535 0.86 AVPR2 (1.00) AVPR2AVPR1A
SCHEMBL8560580 0.85 AVPR2 (0.56) AVPR2AVPR1AALDH1A1
SCHEMBL8563344 0.83 AVPR2 (0.81) AVPR2AVPR1A
SCHEMBL8557743 0.83 AVPR2 (0.64) AVPR2AVPR1AACHE
SCHEMBL8561097 0.83 AVPR2 (0.52) AVPR2AVPR1AHDAC1HDAC8HDAC6
SCHEMBL8557275 0.82 AVPR2 (0.59) AVPR2AVPR1A
SCHEMBL8561645 0.81 AVPR2 (0.58) AVPR2AVPR1AKDM4EACHE
SCHEMBL8558085 0.81 AVPR2 (0.61) AVPR2AVPR1AALDH1A1
SCHEMBL8556252 0.80 NAMPT (0.63) AVPR2AVPR1AKDM4EALDH1A1
SCHEMBL8562554 0.79 AVPR2 (0.73) AVPR2AVPR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640592-B1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID CO (US) 1998-12-30 EP disclosed