SCHEMBL8561645

SCHEMBL8561645

O=C(Nc1ccc(Cl)cc1Cl)c1ccc(C(=O)N2Cc3ccccc3Cc3ccccc32)cc1

nearest known ligand 0.58

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 4/20 0.58
AVPR1A P37288 4/20 0.58
KDM4E B2RXH2 1/20 0.54
NPSR1 Q6W5P4 1/20 0.54
RXFP1 Q9HBX9 1/20 0.54
TAS1R3 Q7RTX0 2/20 0.53
TAS1R1 Q7RTX1 2/20 0.53
TAS1R2 Q8TE23 2/20 0.53
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
ACHE P22303 3/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8559546 0.92 AVPR2 (0.55) AVPR2AVPR1ANPSR1ACHE
SCHEMBL8557607 0.89 NPC1 (0.50) AVPR2AVPR1ANPSR1TAS1R3TAS1R1
SCHEMBL8561097 0.85 AVPR2 (0.52) AVPR2AVPR1ANPC1RAB9A
SCHEMBL8557503 0.84 ACHE (0.58) AVPR2AVPR1ANPC1RAB9AACHE
SCHEMBL8563344 0.83 AVPR2 (0.81) AVPR2AVPR1A
SCHEMBL8558027 0.81 AVPR2 (0.69) AVPR2AVPR1A
SCHEMBL8559006 0.81 AVPR2 (0.75) AVPR2AVPR1AKDM4EACHE
SCHEMBL8563565 0.81 NAMPT (0.50) AVPR2AVPR1AKDM4ENPC1RAB9A
SCHEMBL8562097 0.81 AVPR2 (0.49) AVPR2AVPR1ANPSR1TAS1R3TAS1R1
SCHEMBL8559349 0.81 AVPR2 (0.60) AVPR2AVPR1AACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640592-B1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID CO (US) 1998-12-30 EP disclosed