SCHEMBL8559583

SCHEMBL8559583

O=C(c1ccc([N+](=O)[O-])cc1)N1Cc2ccccc2Sc2ccccc21

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 3/20 0.67
HPGD P15428 1/20 0.51
MAPT P10636 4/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
LMNA P02545 2/20 0.47
GAA P10253 2/20 0.47
MAPK1 P28482 2/20 0.47
SNCA P37840 1/20 0.47
P2RX4 Q99571 1/20 0.47
L3MBTL1 Q9Y468 3/20 0.44
ALDH1A1 P00352 2/20 0.43
MEN1 O00255 1/20 0.43
USP2 O75604 1/20 0.43
POLB P06746 1/20 0.43
HTT P42858 1/20 0.43
KMT2A Q03164 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
AVPR2 P30518 1/20 0.43
AVPR1A P37288 1/20 0.43
ACHE P22303 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8556386 0.86 BCHE (0.52) BCHEHPGDMAPTSMN1; SMN2LMNA
SCHEMBL8557987 0.82 AVPR2 (0.53) BCHEHPGDSMN1; SMN2P2RX4ALDH1A1
SCHEMBL7330482 0.81 HPGD (0.54) BCHEHPGDMAPTSMN1; SMN2LMNA
SCHEMBL10490281 0.80 BCHE (1.00) BCHEMAPTSMN1; SMN2LMNAGAA
SCHEMBL7347407 0.78 BCHE (0.59) BCHEHPGDMAPTSMN1; SMN2LMNA
SCHEMBL8557423 0.76 ACHE (0.51) AVPR2AVPR1AACHE
SCHEMBL7348893 0.76 BCHE (0.56) BCHEHPGDMAPTSMN1; SMN2LMNA
SCHEMBL14509685 0.74 HPGD (0.47) BCHEHPGDMAPTLMNAGAA
SCHEMBL31332440 0.74 HSD17B3 (0.68) BCHE
SCHEMBL7340479 0.74 AVPR1A (0.74) AVPR2AVPR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640592-B1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID CO (US) 1998-12-30 EP disclosed
EP-0640592-A1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID COMPANY (US) 1995-03-01 EP disclosed