SCHEMBL8557423

SCHEMBL8557423

O=C(Nc1ccc(C(=O)N2Cc3ccccc3Sc3ccccc32)cc1)c1ccccc1

nearest known ligand 0.75

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.51
HSD17B3 P37058 1/20 0.50
AVPR2 P30518 3/20 0.49
AVPR1A P37288 3/20 0.49
RAB9A P51151 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8556946 0.86 AVPR2 (0.55) AVPR2AVPR1A
SCHEMBL8555591 0.86 AVPR2 (0.53) AVPR2AVPR1A
SCHEMBL8559251 0.86 AVPR2 (0.68) AVPR2AVPR1A
SCHEMBL8558825 0.86 AVPR1A (0.53) AVPR2AVPR1A
SCHEMBL8559312 0.86 AVPR1A (0.55) AVPR2AVPR1A
SCHEMBL8555635 0.85 HSD11B1 (0.47) ACHERAB9A
SCHEMBL8560419 0.83 AVPR2 (0.52) AVPR2AVPR1ARAB9A
SCHEMBL8558605 0.83 AVPR2 (0.57) AVPR2AVPR1A
SCHEMBL8563255 0.83 AVPR2 (0.59) AVPR2AVPR1A
SCHEMBL8562542 0.83 AVPR1A (0.57) AVPR2AVPR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640592-B1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID CO (US) 1998-12-30 EP disclosed
EP-0640592-A1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID COMPANY (US) 1995-03-01 EP disclosed