SCHEMBL8559786

SCHEMBL8559786

Cc1cccc(C(=O)Nc2nc(C)c(C)s2)c1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 10/20 0.74
NPC1 O15118 8/20 0.74
SMN1; SMN2 Q16637 4/20 0.74
PKM P14618 2/20 0.74
SCD O00767 2/20 0.66
MAPT P10636 5/20 0.62
TP53 P04637 1/20 0.62
KMT2A Q03164 6/20 0.57
KDM4E B2RXH2 2/20 0.57
ALDH1A1 P00352 1/20 0.57
LMNA P02545 1/20 0.57
RXFP1 Q9HBX9 2/20 0.57
MEN1 O00255 4/20 0.57
GRM5 P41594 1/20 0.56
CRHBP P24387 1/20 0.56
RECQL P46063 1/20 0.56
CRHR2 Q13324 1/20 0.56
KCNK3 O14649 1/20 0.55
KCNH2 Q12809 1/20 0.55
KCNK9 Q9NPC2 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7349284 0.86 RAB9A (0.70) RAB9ANPC1SMN1; SMN2PKMSCD
SCHEMBL31665475 0.85 NPC1 (1.00) RAB9ANPC1SMN1; SMN2PKMMAPT
SCHEMBL3581515 0.85 RAB9A (0.81) RAB9ANPC1SMN1; SMN2PKMSCD
SCHEMBL2754020 0.82 NPC1 (0.77) RAB9ANPC1SMN1; SMN2PKMMAPT
SCHEMBL14985591 0.80 SCD (0.81) RAB9ANPC1SMN1; SMN2SCDMAPT
SCHEMBL8552971 0.80 SCD (1.00) RAB9ANPC1SMN1; SMN2SCDMAPT
SCHEMBL1969659 0.79 RAB9A (0.64) RAB9ANPC1SMN1; SMN2PKMMAPT
SCHEMBL4917918 0.79 SCD (0.67) RAB9ANPC1SMN1; SMN2SCDMAPT
SCHEMBL8556554 0.78 KMT2A (0.75) RAB9ANPC1SMN1; SMN2SCDMAPT
SCHEMBL8117715 0.78 RAB9A (0.70) RAB9ANPC1SMN1; SMN2PKMMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0815108-A1 CYCLIC UREA HIV PROTEASE INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1998-01-07 EP claimed
US-5683999-A Cyclic urea HIV protease inhibitors THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1997-11-04 US claimed
EP-0815108-A1 CYCLIC UREA HIV PROTEASE INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1998-01-07 EP disclosed
US-5683999-A Cyclic urea HIV protease inhibitors THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1997-11-04 US disclosed