SCHEMBL8560147

SCHEMBL8560147

CCOC(=O)c1cnc2nc(C=CC(=O)O)c(OCC)cc2c1O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 8/20 0.42
ALDH1A1 P00352 3/20 0.37
MAPT P10636 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
LMNA P02545 1/20 0.37
MAPK1 P28482 1/20 0.37
ATM Q13315 1/20 0.37
TSHR P16473 1/20 0.36
KDM4E B2RXH2 3/20 0.36
GAA P10253 2/20 0.36
NPC1 O15118 1/20 0.36
TP53 P04637 1/20 0.36
RAB9A P51151 1/20 0.36
KMT2A Q03164 1/20 0.36
THRB P10828 1/20 0.36
CCNB2 O95067 1/20 0.36
CDK1 P06493 1/20 0.36
CCNB1 P14635 1/20 0.36
CCNA2 P20248 1/20 0.36
CCNE1 P24864 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8560142 1.00 DPP4 (0.42) DPP4ALDH1A1MAPTSMN1; SMN2LMNA
SCHEMBL8322260 0.81 DPP4 (0.48) DPP4MAPTTSHRKDM4ENPC1
SCHEMBL8565165 0.81 PDE4B (0.52) ALDH1A1MAPTSMN1; SMN2GAATP53
SCHEMBL8565169 0.81 PDE4B (0.52) ALDH1A1MAPTSMN1; SMN2GAATP53
SCHEMBL8558995 0.81 DPP4 (0.46) DPP4ALDH1A1MAPTSMN1; SMN2LMNA
Hydrochloric Acid SCHEMBL8327789 0.80 PDE4B (0.51) ALDH1A1MAPTSMN1; SMN2GAATP53
SCHEMBL8324234 0.74 DPP4 (0.51) DPP4MAPTSMN1; SMN2LMNATSHR
SCHEMBL8324245 0.73 TSHR (0.42) DPP4ALDH1A1MAPTSMN1; SMN2LMNA
SCHEMBL8325264 0.72 PDE4B (0.51) ALDH1A1MAPTSMN1; SMN2GAATP53
SCHEMBL8327280 0.72 PDE4B (0.51) ALDH1A1MAPTSMN1; SMN2GAATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0618916-B1 ANTI-RHEUMATIC NAPHTHYRIDINE DERIVATIVES KNOLL AG (DE) 1998-09-23 EP disclosed
US-5464781-A TREATING RHEUMATIC DISEASES THE BOOTS COMPANY PLC (GB) 1995-11-07 US disclosed
WO-1993013097-A1 ANTI-RHEUMATIC NAPHTHYRIDINE DERIVATIVES THE BOOTS COMPANY PLC (GB) 1993-07-08 WO disclosed