SCHEMBL8560359

SCHEMBL8560359

CCCCCCc1cc(CCCCCC)cc(CCCCCC)c1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 5/20 0.70
CYP3A4 P08684 2/20 0.65
GPR84 Q9NQS5 2/20 0.61
ESR1 P03372 2/20 0.56
ADRA2A P08913 2/20 0.56
ADORA3 P0DMS8 2/20 0.56
TACR2 P21452 2/20 0.56
SLC6A2 P23975 2/20 0.56
SLC6A4 P31645 2/20 0.56
SLC6A3 Q01959 2/20 0.56
KDM4E B2RXH2 1/20 0.56
ALDH1A1 P00352 1/20 0.56
LMNA P02545 1/20 0.56
SHBG P04278 1/20 0.56
TP53 P04637 1/20 0.56
HSPD1 P10809 1/20 0.56
ADRB3 P13945 1/20 0.56
HTR2C P28335 1/20 0.56
HSPE1 P61604 1/20 0.56
HIF1A Q16665 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7628223 1.00 PTGS2 (0.70) PTGS2CYP3A4GPR84ESR1ADRA2A
SCHEMBL9122379 1.00 PTGS2 (0.70) PTGS2CYP3A4GPR84ESR1ADRA2A
SCHEMBL9420945 0.97 PTGS2 (0.67) PTGS2CYP3A4GPR84ESR1ADRA2A
SCHEMBL2871788 0.97 PTGS2 (0.68) PTGS2CYP3A4GPR84ESR1ADRA2A
Ethylene SCHEMBL28058312 0.95 PTGS2 (0.64) PTGS2CYP3A4GPR84ESR1ADRA2A
SCHEMBL1187883 0.92 PTGS2 (0.61) PTGS2CYP3A4GPR84ESR1ADRA2A
SCHEMBL1187238 0.92 PTGS2 (0.61) PTGS2CYP3A4GPR84ESR1ADRA2A
SCHEMBL1186501 0.92 PTGS2 (0.61) PTGS2CYP3A4GPR84ESR1ADRA2A
SCHEMBL1187931 0.92 PTGS2 (0.61) PTGS2CYP3A4GPR84ESR1ADRA2A
SCHEMBL1186551 0.92 PTGS2 (0.61) PTGS2CYP3A4GPR84ESR1ADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113200812-B 1,3,5-trisubstituted aryl compound synthesis method 天津大学 2023-04-07 CN disclosed
CN-113200812-A Synthesis method of 1,3, 5-trisubstituted aryl compound 天津大学 2021-08-03 CN disclosed
US-5756730-A Process for preparing analgesic compounds SANKYO COMPANY, LIMITED (JP) 1998-05-26 US disclosed
US-5656758-A AMIDATION OF AN AMINE-CONTAINING THIOMORPHOLINE OR PIPERAZINE COMPOUND SANKYO COMPANY, LIMITED (JP) 1997-08-12 US disclosed
US-5512567-A KAPPA-RECEPTOR AGONISTS SANKYO COMPANY, LIMITED (JP) 1996-04-30 US disclosed
US-5385721-A X-ray radiology and computer tomography; uniform coating of the soft tissues; medical diagnosis STERLING WINTHROP INC. (US) 1995-01-31 US disclosed
EP-0609589-A2 Compositions of alkylbenzenes in film-forming materials for visualization of the gastrointestinal tract NYCOMED IMAGING AS (NO) 1994-08-10 EP disclosed
EP-0609588-A2 Compositions of alkylbenzenes for visualization of the gastrointestinal tract NYCOMED IMAGING AS (NO) 1994-08-10 EP disclosed
US-5334370-A X-ray contrast mixtures for diagnostic radiology consisting of iodo alkylbenzene, a polysaccharide salt or a anionic polymers STERLING WINTHROP INC. (US) 1994-08-02 US disclosed
US-5308607-A FOR USE IN DIAGNOSTIC RADIOLOGY STERLING WINTHROP INC. (US) 1994-05-03 US disclosed
US-5270327-A Piperidine derivatives SANKYO COMPANY, LIMITED (JP) 1993-12-14 US disclosed
EP-0356247-B1 ANALGESIC CARBOXYLIC ACID AMIDE DERIVATIVES Sankyo Company Limited (JP) 1993-03-17 EP disclosed
US-5021413-A Analgesic thiomorpholins their preparation, and pharmaceutical compositions containing them SANKYO COMPANY LIMITED (JP) 1991-06-04 US disclosed
EP-0207737-B1 PROCESS FOR THE STABILIZATION OF MERCAPTOBENZOTHIAZOLE IN A LUBRICATING OIL COMPOSITION EXXON RESEARCH AND ENGINEERING COMPANY (US) 1990-12-19 EP disclosed
EP-0356247-A1 Analgesic carboxylic acid amide derivatives Sankyo Company Limited (JP) 1990-02-28 EP disclosed
EP-0207737-A2 Process for the stabilization of mercaptobenzothiazole in a lubricating oil composition EXXON RESEARCH AND ENGINEERING COMPANY (US) 1987-01-07 EP disclosed
US-4589991-A FORMING AN AMINE SALT OF MERCAPTOBENZOTHIAZOLE, DISSOLVING IN AROMATIC ETHER SOLVENT EXXON RESEARCH & ENGINEERING CO. (US) 1986-05-20 US disclosed