SCHEMBL8560515

SCHEMBL8560515

CCOC(=O)CCc1ccc(N2CCN(c3ccc4c(c3)CCN(C)CC4)C2=O)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP4F2 P78329 1/20 0.45
CYP4A11 Q02928 1/20 0.45
TMEM97 Q5BJF2 5/20 0.43
SIGMAR1 Q99720 5/20 0.43
SLC6A2 P23975 2/20 0.43
HRH2 P25021 2/20 0.43
HRH1 P35367 2/20 0.43
CHRM5 P08912 2/20 0.43
HTR2A P28223 2/20 0.43
HTR2C P28335 2/20 0.43
HTR1A P08908 1/20 0.43
ADRA1D P25100 1/20 0.43
HTR1B P28222 1/20 0.43
HTR1E P28566 1/20 0.43
HTR2B P41595 1/20 0.43
SLC6A3 Q01959 1/20 0.43
HRH3 Q9Y5N1 2/20 0.43
S1PR1 P21453 1/20 0.41
CHRM1 P11229 2/20 0.39
MEN1 O00255 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8563637 0.99 CYP4F2 (0.44) CYP4F2CYP4A11TMEM97SIGMAR1SLC6A2
SCHEMBL8559518 0.89 HRH3 (0.41) TMEM97SIGMAR1CHRM5HTR2AHTR2C
Hydrochloric Acid SCHEMBL8564996 0.88 HRH3 (0.40) TMEM97SIGMAR1CHRM5HTR2AHTR2C
SCHEMBL8565812 0.86 NOTUM (0.39) CYP4F2CYP4A11TMEM97SIGMAR1HTR2A
SCHEMBL8559863 0.85 S1PR1 (0.50) TMEM97SIGMAR1HTR2AHTR2CHRH3
Hydrochloric Acid SCHEMBL8559741 0.85 NOTUM (0.38) CYP4F2CYP4A11TMEM97SIGMAR1HTR2A
Hydrochloric Acid SCHEMBL8563445 0.84 S1PR1 (0.49) TMEM97SIGMAR1HTR2AHTR2CHRH3
SCHEMBL8559326 0.83 S1PR1 (0.47) TMEM97SIGMAR1HRH3S1PR1DRD2
SCHEMBL8562720 0.81 S1PR1 (0.45) TMEM97SIGMAR1SLC6A2HRH2HRH1
SCHEMBL7390478 0.81 CYP4F2 (0.52) CYP4F2CYP4A11HRH3S1PR1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0612741-B1 Cyclic derivatives, medicaments containing them and process for their preparation THOMAE GMBH DR K (DE) 1998-06-10 EP claimed
EP-0612741-A1 Cyclic derivatives, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1994-08-31 EP claimed
US-5827849-A HAVING INHIBITORY EFFECT ON INFLAMMATION AND BONE DEGRADATION, ANTITHROMBOTIC, ANTIAGGREGATORY AND TUMOR- OR METASTASIS-INHIBITING EFFECT KARL THOMAE GMBH (DE) 1998-10-27 US disclosed
EP-0612741-B1 Cyclic derivatives, medicaments containing them and process for their preparation THOMAE GMBH DR K (DE) 1998-06-10 EP disclosed
US-5612335-A ANTICOAGULANTS; COMBATING/PREVENTING DISEASES WHERE CELL AGGREGATES OCCUR OR CELL-MATRIX INTERACTIONS PLAY A PART KARL THOMAE GMBH (DE) 1997-03-18 US disclosed
US-5519036-A IMIDAZOLIDINONES, ANTICOAGULANTS, CELL AGGREGATION PREVENTION KARL THOMAE GMBH (DE) 1996-05-21 US disclosed
EP-0612741-A1 Cyclic derivatives, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1994-08-31 EP disclosed