SCHEMBL8565812

SCHEMBL8565812

CC(C)OC(=O)CCc1ccc(N2CCN(c3ccc4c(c3)CCN(C)CC4)C2=O)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.39
S1PR1 P21453 2/20 0.39
FAAH O00519 3/20 0.37
DRD2 P14416 2/20 0.37
DRD3 P35462 2/20 0.37
KCNH2 Q12809 1/20 0.37
MAPT P10636 2/20 0.35
ALOX15 P16050 2/20 0.35
CASP1 P29466 2/20 0.35
CASP7 P55210 2/20 0.35
HSD17B10 Q99714 2/20 0.35
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35
USP2 O75604 1/20 0.35
ALDH1A1 P00352 1/20 0.35
POLB P06746 1/20 0.35
THRB P10828 1/20 0.35
BRCA1 P38398 1/20 0.35
RECQL P46063 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8559741 0.99 NOTUM (0.38) NOTUMS1PR1FAAHDRD2DRD3
SCHEMBL8558614 0.90 HTR6 (0.38) NOTUMS1PR1FAAHDRD2DRD3
Hydrochloric Acid SCHEMBL8568700 0.89 HTR6 (0.38) NOTUMS1PR1FAAHDRD2DRD3
SCHEMBL8559518 0.88 HRH3 (0.41) NOTUMS1PR1DRD2DRD3POLB
Hydrochloric Acid SCHEMBL8564996 0.87 HRH3 (0.40) S1PR1DRD2DRD3POLBTMEM97
SCHEMBL8560515 0.86 CYP4F2 (0.45) NOTUMS1PR1DRD2DRD3MEN1
Hydrochloric Acid SCHEMBL8563637 0.85 CYP4F2 (0.44) NOTUMS1PR1DRD2DRD3MEN1
SCHEMBL8559863 0.85 S1PR1 (0.50) S1PR1DRD2DRD3ALDH1A1L3MBTL1
Hydrochloric Acid SCHEMBL8563445 0.84 S1PR1 (0.49) S1PR1DRD2DRD3ALDH1A1L3MBTL1
SCHEMBL8559326 0.82 S1PR1 (0.47) S1PR1DRD2DRD3ALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0612741-B1 Cyclic derivatives, medicaments containing them and process for their preparation THOMAE GMBH DR K (DE) 1998-06-10 EP claimed
EP-0612741-A1 Cyclic derivatives, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1994-08-31 EP claimed
US-5827849-A HAVING INHIBITORY EFFECT ON INFLAMMATION AND BONE DEGRADATION, ANTITHROMBOTIC, ANTIAGGREGATORY AND TUMOR- OR METASTASIS-INHIBITING EFFECT KARL THOMAE GMBH (DE) 1998-10-27 US disclosed
EP-0612741-B1 Cyclic derivatives, medicaments containing them and process for their preparation THOMAE GMBH DR K (DE) 1998-06-10 EP disclosed
US-5612335-A ANTICOAGULANTS; COMBATING/PREVENTING DISEASES WHERE CELL AGGREGATES OCCUR OR CELL-MATRIX INTERACTIONS PLAY A PART KARL THOMAE GMBH (DE) 1997-03-18 US disclosed
US-5519036-A IMIDAZOLIDINONES, ANTICOAGULANTS, CELL AGGREGATION PREVENTION KARL THOMAE GMBH (DE) 1996-05-21 US disclosed
EP-0612741-A1 Cyclic derivatives, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1994-08-31 EP disclosed