SCHEMBL8559518

SCHEMBL8559518

COC(=O)CCc1ccc(N2CCN(c3ccc4c(c3)CCN(C)CC4)C2=O)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.41
S1PR1 P21453 2/20 0.40
TMEM97 Q5BJF2 2/20 0.38
SIGMAR1 Q99720 2/20 0.38
DRD2 P14416 3/20 0.38
DRD3 P35462 3/20 0.38
HTR6 P50406 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
HTR2A P28223 1/20 0.38
HTR2C P28335 1/20 0.38
CYP2C19 P33261 1/20 0.38
HDAC1 Q13547 2/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
POLB P06746 1/20 0.36
ABCB1 P08183 1/20 0.36
ABCG2 Q9UNQ0 1/20 0.36
GRIN1 Q05586 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8564996 0.99 HRH3 (0.40) HRH3S1PR1TMEM97SIGMAR1DRD2
SCHEMBL8560515 0.89 CYP4F2 (0.45) HRH3S1PR1TMEM97SIGMAR1DRD2
SCHEMBL8559578 0.89 HTR6 (0.42) HRH3S1PR1DRD2DRD3HTR6
SCHEMBL8562720 0.89 S1PR1 (0.45) HRH3S1PR1TMEM97SIGMAR1DRD2
SCHEMBL8565812 0.88 NOTUM (0.39) S1PR1TMEM97SIGMAR1DRD2DRD3
Hydrochloric Acid SCHEMBL8566255 0.88 HTR6 (0.41) HRH3S1PR1DRD2DRD3HTR6
Hydrochloric Acid SCHEMBL8563637 0.88 CYP4F2 (0.44) HRH3S1PR1TMEM97SIGMAR1DRD2
SCHEMBL8559863 0.87 S1PR1 (0.50) HRH3S1PR1TMEM97SIGMAR1DRD2
Hydrochloric Acid SCHEMBL8559741 0.87 NOTUM (0.38) S1PR1TMEM97SIGMAR1DRD2DRD3
Hydrochloric Acid SCHEMBL8563445 0.86 S1PR1 (0.49) HRH3S1PR1TMEM97SIGMAR1DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0612741-B1 Cyclic derivatives, medicaments containing them and process for their preparation THOMAE GMBH DR K (DE) 1998-06-10 EP claimed
EP-0612741-A1 Cyclic derivatives, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1994-08-31 EP claimed
US-5827849-A HAVING INHIBITORY EFFECT ON INFLAMMATION AND BONE DEGRADATION, ANTITHROMBOTIC, ANTIAGGREGATORY AND TUMOR- OR METASTASIS-INHIBITING EFFECT KARL THOMAE GMBH (DE) 1998-10-27 US disclosed
US-5612335-A ANTICOAGULANTS; COMBATING/PREVENTING DISEASES WHERE CELL AGGREGATES OCCUR OR CELL-MATRIX INTERACTIONS PLAY A PART KARL THOMAE GMBH (DE) 1997-03-18 US disclosed
US-5519036-A IMIDAZOLIDINONES, ANTICOAGULANTS, CELL AGGREGATION PREVENTION KARL THOMAE GMBH (DE) 1996-05-21 US disclosed
EP-0612741-A1 Cyclic derivatives, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1994-08-31 EP disclosed