SCHEMBL8560583

SCHEMBL8560583

O=C1C(Br)CCN1c1ccccc1F

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.53
MEN1 O00255 2/20 0.53
FPR2 P25090 1/20 0.44
NOTUM Q6P988 1/20 0.41
MGLL Q99685 1/20 0.41
GRM2 Q14416 1/20 0.37
LMNA P02545 1/20 0.37
ALDH1A1 P00352 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
TSHR P16473 2/20 0.37
KDM4E B2RXH2 1/20 0.37
POLB P06746 1/20 0.37
HSD11B1 P28845 1/20 0.37
HSD17B10 Q99714 1/20 0.36
OPRM1 P35372 1/20 0.36
KCNH2 Q12809 1/20 0.36
SIGMAR1 Q99720 1/20 0.36
P2RX7 Q99572 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8560584 1.00 KMT2A (0.53) KMT2AMEN1FPR2NOTUMMGLL
SCHEMBL28437828 0.80 HDAC1 (0.48) NOTUMMGLLALDH1A1KDM4EHSD11B1
SCHEMBL6860135 0.80 CCR1 (0.39) LMNAALDH1A1SMN1; SMN2TSHROPRM1
SCHEMBL8567665 0.78 ATM (0.58) KMT2AMEN1MGLLLMNAALDH1A1
SCHEMBL8564613 0.78 ALDH1A1 (0.46) KMT2AMEN1LMNAALDH1A1TSHR
SCHEMBL8567660 0.78 ATM (0.58) KMT2AMEN1MGLLLMNAALDH1A1
SCHEMBL8564617 0.78 ALDH1A1 (0.46) KMT2AMEN1LMNAALDH1A1TSHR
SCHEMBL892631 0.76 NOTUM (0.51) KMT2AMEN1FPR2NOTUMLMNA
SCHEMBL1514921 0.75 MEN1 (0.50) KMT2AMEN1FPR2MGLLALDH1A1
SCHEMBL12285262 0.75 KMT2A (0.47) KMT2AMEN1FPR2NOTUMMGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1060778-C Cephalosporin derivatives HOFFMANN LA ROCHE (CH) 2001-01-17 CN disclosed
US-5804577-A ANTIBIOTICS HOFFMANN-LA ROCHE INC. (US) 1998-09-08 US disclosed
CN-1150950-A Cephalosporin derivatives HOFFMANN LA ROCHE (CH) 1997-06-04 CN disclosed
EP-0761673-A1 Cephalosporin derivatives F. HOFFMANN-LA ROCHE AG (CH) 1997-03-12 EP disclosed