SCHEMBL8560714

SCHEMBL8560714

O=C(N1CCc2ccc(N3CCNS3(=O)=O)cc2CC1)C(F)(F)F

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 7/20 0.47
ESR2 Q92731 7/20 0.47
HDAC6 Q9UBN7 2/20 0.37
PKM P14618 1/20 0.36
ABHD6 Q9BV23 7/20 0.35
HDAC8 Q9BY41 1/20 0.32
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA7 P43166 1/20 0.32
CA9 Q16790 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL373697 0.72 ESR2 (0.83) ESR1ESR2HDAC6ABHD6CA1
SCHEMBL566629 0.71 ESR1 (0.58) ESR1ESR2HDAC6PKMABHD6
SCHEMBL2585109 0.71 ESR1 (0.62) ESR1ESR2HDAC6PKMABHD6
SCHEMBL373718 0.71 ESR1 (0.58) ESR1ESR2HDAC6PKMABHD6
SCHEMBL7849236 0.71 ESR2 (0.58) ESR1ESR2HDAC6PKMABHD6
SCHEMBL1787936 0.71 ABHD6 (0.60) ESR1ESR2HDAC6PKMABHD6
SCHEMBL27176737 0.71 ESR1 (0.58) ESR1ESR2HDAC6PKMABHD6
SCHEMBL1791230 0.70 ESR1 (0.55) ESR1ESR2HDAC6PKM
SCHEMBL7423258 0.70 ESR1 (0.57) ESR1ESR2HDAC6PKMABHD6
SCHEMBL506139 0.70 ESR1 (0.59) ESR1ESR2ABHD6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5827849-A HAVING INHIBITORY EFFECT ON INFLAMMATION AND BONE DEGRADATION, ANTITHROMBOTIC, ANTIAGGREGATORY AND TUMOR- OR METASTASIS-INHIBITING EFFECT KARL THOMAE GMBH (DE) 1998-10-27 US disclosed
US-5612335-A ANTICOAGULANTS; COMBATING/PREVENTING DISEASES WHERE CELL AGGREGATES OCCUR OR CELL-MATRIX INTERACTIONS PLAY A PART KARL THOMAE GMBH (DE) 1997-03-18 US disclosed
US-5519036-A IMIDAZOLIDINONES, ANTICOAGULANTS, CELL AGGREGATION PREVENTION KARL THOMAE GMBH (DE) 1996-05-21 US disclosed