SCHEMBL8560716

SCHEMBL8560716

COCCOc1cnc2ccccc2c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.49
CYP1A2 P05177 1/20 0.49
KDM4E B2RXH2 4/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
KMT2A Q03164 1/20 0.48
PDGFRB P09619 3/20 0.47
PDGFRA P16234 3/20 0.47
CHRNB2 P17787 2/20 0.46
CHRNA4 P43681 1/20 0.46
KDM1A O60341 2/20 0.44
MAPK1 P28482 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
RAB9A P51151 2/20 0.42
MET P08581 1/20 0.42
NPC1 O15118 1/20 0.40
ALDH1A1 P00352 1/20 0.40
MAPT P10636 1/20 0.40
HPGD P15428 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
CHRNB1 P11230 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23412249 0.86 KDM4E (0.59) CYP1A2KDM4ESMN1; SMN2KMT2APDGFRB
SCHEMBL23413027 0.86 KDM4E (0.59) CYP1A2KDM4ESMN1; SMN2KMT2APDGFRB
SCHEMBL8564487 0.85 CYP1A2 (0.50) CYP1A2KDM4ESMN1; SMN2KMT2APDGFRB
SCHEMBL8566047 0.85 TLR8 (0.54) CYP1A2KDM4ESMN1; SMN2KMT2APDGFRB
SCHEMBL16836341 0.83 RAB9A (0.57) CYP1A2KDM4ESMN1; SMN2KMT2APDGFRB
SCHEMBL13533394 0.82 TLR8 (0.58) CYP1A2KDM4ESMN1; SMN2KMT2APDGFRB
SCHEMBL16836548 0.82 TLR8 (0.56) TSHRCYP1A2KDM4ESMN1; SMN2KMT2A
SCHEMBL29935791 0.81 PDGFRB (0.49) CYP1A2KDM4ESMN1; SMN2KMT2APDGFRB
SCHEMBL30898597 0.81 RAB9A (0.50) CYP1A2KDM4ESMN1; SMN2KMT2APDGFRB
SCHEMBL29248551 0.81 RAB9A (0.50) CYP1A2KDM4ESMN1; SMN2KMT2APDGFRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102958918-B Novel tobacco amide derivatives or its salt FUJIFILM CORP. (JP) 2015-12-09 CN disclosed
CN-103492377-A Triazolopyridine compounds as PIM kinase inhibitors ARRAY BIOPHARMA INC 2014-01-01 CN disclosed
US-5719141-A HYPOTENSIVE AGENTS NOVARTIS CORPORATION (US) 1998-02-17 US disclosed
CN-1169986-A 2.9-diamino-and 2-amino-8-carbamoyl-4-hydroxy-aldanoic acid amide derivatives CIBA GEIGY AG (CH) 1998-01-14 CN disclosed
EP-0702004-A2 2,9-diamino- and 2-amino-8-carbamoyl-4-hydroxy-alkanoic acid amid derivatives CIBA-GEIGY AG (CH) 1996-03-20 EP disclosed