SCHEMBL8560971

SCHEMBL8560971

COc1ccc(CN2C(=O)C(N)C(=O)N(CCC(C)C)c3ccccc32)cc1

nearest known ligand 0.53

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 2/20 0.50
CASP3 P42574 1/20 0.46
CMA1 P23946 1/20 0.46
GSK3B P49841 3/20 0.45
ADK P55263 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
GSK3A P49840 1/20 0.44
ALDH1A1 P00352 1/20 0.43
HTT P42858 1/20 0.43
TSHR P16473 2/20 0.42
LMNA P02545 1/20 0.42
SIRT2 Q8IXJ6 1/20 0.42
SIRT1 Q96EB6 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7754062 0.80 CMA1 (0.47) CCKBRCASP3CMA1GSK3BADK
SCHEMBL8563195 0.79 CCKBR (0.84) CCKBR
SCHEMBL8405020 0.77 CCKAR (0.56) CCKBR
SCHEMBL8866387 0.76 CCKBR (0.48) CCKBRALDH1A1
SCHEMBL4429210 0.76 GSK3B (0.52) CASP3CMA1GSK3BADKL3MBTL1
SCHEMBL3173671 0.76 GSK3B (0.52) CASP3CMA1GSK3BADKL3MBTL1
SCHEMBL4422395 0.76 GSK3B (0.52) CASP3CMA1GSK3BADKL3MBTL1
SCHEMBL8559078 0.76 BACE1 (0.50) CCKBRCMA1GSK3BADKL3MBTL1
Hydrochloric Acid SCHEMBL3854466 0.75 GSK3B (0.51) CASP3CMA1GSK3BADKL3MBTL1
SCHEMBL8547144 0.74 CCKBR (0.60) CCKBR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5716953-A MODIFIERS OF GASTRIN AND CHOLECYSTOKININS GLAXO WELLCOME S.P.A. (IT) 1998-02-10 US disclosed