SCHEMBL8561220

SCHEMBL8561220

O=C1NCC(c2ccc(Cl)c(Cl)c2)CC1CCCOC1CCCCO1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
SLC6A2 P23975 10/20 0.37
SLC6A3 Q01959 10/20 0.37
SLC6A4 P31645 4/20 0.37
CYP2D6 P10635 1/20 0.37
KCNH2 Q12809 1/20 0.37
PTAFR P25105 3/20 0.36
PDE4D Q08499 2/20 0.35
KDM4C Q9H3R0 1/20 0.33
KCNA5 P22460 1/20 0.32
SCN5A Q14524 1/20 0.32
NAAA Q02083 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8558084 0.78 PTAFR (0.37) MEN1KMT2APTAFRPDE4DKDM4C
SCHEMBL8291780 0.71 KCNH2 (0.48) MEN1KMT2ASLC6A2SLC6A3SLC6A4
SCHEMBL8366968 0.69 PTAFR (0.39) SLC6A2SLC6A3SLC6A4CYP2D6KCNH2
SCHEMBL8478669 0.69 PTAFR (0.39) SLC6A2SLC6A3SLC6A4CYP2D6KCNH2
SCHEMBL8307213 0.68 PTAFR (0.34) SLC6A2SLC6A3SLC6A4CYP2D6KCNH2
SCHEMBL8564881 0.67 PDE4A (0.38) MEN1KMT2APDE4DKDM4CKCNA5
SCHEMBL7956526 0.67 MEN1 (0.38) MEN1KMT2ASLC6A2SLC6A3SLC6A4
SCHEMBL8702363 0.66 MEN1 (0.37) MEN1KMT2ASLC6A2SLC6A3SLC6A4
SCHEMBL4630820 0.65 MEN1 (0.39) MEN1KMT2ASLC6A2SLC6A3SLC6A4
SCHEMBL11148815 0.65 MEN1 (0.45) MEN1KMT2AKDM4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5807865-A 3,3-disubstituted piperidine derivatives and their use as therapeutic agents MERCK SHARP & DOHME LIMITED (GB) 1998-09-15 US disclosed