SCHEMBL8558084

SCHEMBL8558084

O=C1C(CCCOC2CCCCO2)CC(c2ccc(Cl)c(Cl)c2)CN1Cc1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTAFR P25105 2/20 0.37
PDE4A P27815 3/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
PDE4B Q07343 1/20 0.35
PDE4C Q08493 1/20 0.35
PDE4D Q08499 1/20 0.35
TACR1 P25103 3/20 0.34
P2RX3 P56373 4/20 0.34
KDM4C Q9H3R0 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8564881 0.87 PDE4A (0.38) PDE4AMEN1KMT2APDE4BPDE4C
SCHEMBL8558380 0.79 HPGD (0.40) PDE4APDE4BPDE4CPDE4DTACR1
SCHEMBL8561168 0.79 PDE4A (0.40) PDE4APDE4BPDE4CPDE4DTACR1
SCHEMBL8561220 0.78 MEN1 (0.39) PTAFRMEN1KMT2APDE4DKDM4C
Hydrochloric Acid SCHEMBL8593049 0.71 CCR3 (0.42) MEN1KMT2ATACR1
SCHEMBL8707339 0.71 TACR1 (0.43) PDE4AMEN1KMT2APDE4BPDE4C
SCHEMBL7846541 0.71 TACR1 (0.60) TACR1
SCHEMBL8291780 0.71 KCNH2 (0.48) PTAFRMEN1KMT2A
SCHEMBL4631281 0.69 TACR1 (0.45) TACR1
SCHEMBL8300796 0.69 TACR1 (0.59) TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5807865-A 3,3-disubstituted piperidine derivatives and their use as therapeutic agents MERCK SHARP & DOHME LIMITED (GB) 1998-09-15 US disclosed