SCHEMBL8562729

SCHEMBL8562729

COC(=O)C(COCc1ccccc1)(OCC1(c2ccccc2)CCN(C(=O)OC(C)(C)C)CC1)c1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.70

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 20/20 0.70
SLC6A4 P31645 6/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5216125 0.83 TACR1 (1.00) TACR1SLC6A4
SCHEMBL8561630 0.79 TACR1 (0.67) TACR1SLC6A4
SCHEMBL13404344 0.77 TACR1 (0.88) TACR1SLC6A4
SCHEMBL13404342 0.77 TACR1 (0.88) TACR1SLC6A4
SCHEMBL3594793 0.77 TACR1 (0.88) TACR1SLC6A4
SCHEMBL13404345 0.76 TACR1 (0.82) TACR1SLC6A4
SCHEMBL13404343 0.76 TACR1 (0.82) TACR1SLC6A4
SCHEMBL8545581 0.75 TACR1 (0.72) TACR1SLC6A4
SCHEMBL14541562 0.75 TACR1 (0.84) TACR1SLC6A4
SCHEMBL8546545 0.75 TACR1 (0.66) TACR1SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5760018-A Gem-disubstituted azacyclic tachykinin antagonists MERCK SHARP & DOHME LTD. (GB) 1998-06-02 US disclosed
WO-1995019344-A1 GEM-DISUBSTITUTED AZACYCLIC TACHYKININ ANTAGONISTS MERCK SHARP & DOHME LIMITED (GB) 1995-07-20 WO disclosed