SCHEMBL8561673

SCHEMBL8561673

CCOC(=O)N1CNc2ccccc2C1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.51
BRD4 O60885 1/20 0.49
ALDH1A1 P00352 3/20 0.44
HSP90AA1 P07900 1/20 0.44
MAPT P10636 4/20 0.44
RAB9A P51151 2/20 0.44
MEN1 O00255 1/20 0.44
MDM2 Q00987 1/20 0.44
KMT2A Q03164 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
NOS2 P35228 1/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
LMNA P02545 2/20 0.43
GAA P10253 4/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
TSHR P16473 1/20 0.43
NAMPT P43490 1/20 0.42
NPC1 O15118 1/20 0.42
CYP2C9 P11712 1/20 0.42
ALOX15 P16050 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6677698 0.81 NOTUM (0.57) MAPK1ALDH1A1HSP90AA1MAPTRAB9A
SCHEMBL27993916 0.78 MAPK1 (0.48) MAPK1BRD4HSP90AA1MAPTRAB9A
SCHEMBL28126317 0.77 MAPK1 (0.41) MAPK1ALDH1A1NAMPT
SCHEMBL28413210 0.76 MAPK1 (0.47) MAPK1BRD4HSP90AA1MAPTMEN1
SCHEMBL4880946 0.76 BRD4 (0.45) MAPK1BRD4ALDH1A1HSP90AA1MAPT
SCHEMBL16268868 0.74 ALDH1A1 (0.64) MAPK1ALDH1A1MAPTRAB9AMEN1
SCHEMBL14149488 0.73 MAPK1 (0.43) MAPK1BRD4ALDH1A1MAPTMEN1
SCHEMBL3089343 0.73 SMN1; SMN2 (0.46) MAPK1BRD4ALDH1A1MAPTRAB9A
SCHEMBL3149403 0.71 MAPK1 (0.62) MAPK1RAB9AMEN1KMT2ANPSR1
SCHEMBL1295044 0.71 ALDH1A1 (0.64) ALDH1A1MAPTMEN1KMT2AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5719141-A HYPOTENSIVE AGENTS NOVARTIS CORPORATION (US) 1998-02-17 US disclosed
CN-1169986-A 2.9-diamino-and 2-amino-8-carbamoyl-4-hydroxy-aldanoic acid amide derivatives CIBA GEIGY AG (CH) 1998-01-14 CN disclosed
EP-0702004-A2 2,9-diamino- and 2-amino-8-carbamoyl-4-hydroxy-alkanoic acid amid derivatives CIBA-GEIGY AG (CH) 1996-03-20 EP disclosed