SCHEMBL8562028

SCHEMBL8562028

Cc1ccc(C(=CS(=O)(=O)Cl)c2ccccc2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.55
L3MBTL1 Q9Y468 2/20 0.55
CYP1A2 P05177 1/20 0.55
CYP2C9 P11712 1/20 0.55
CYP2C19 P33261 1/20 0.55
NPSR1 Q6W5P4 1/20 0.55
MCOLN3 Q8TDD5 1/20 0.55
PTGS2 P35354 4/20 0.53
CES2 O00748 1/20 0.50
CES1 P23141 1/20 0.50
MEN1 O00255 1/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
KMT2A Q03164 1/20 0.46
LMNA P02545 3/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
NOD2 Q9HC29 1/20 0.46
RECQL P46063 1/20 0.42
HSD11B1 P28845 1/20 0.42
POLB P06746 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7372442 0.89 ALDH1A1 (0.61) ALDH1A1L3MBTL1CYP1A2CYP2C9CYP2C19
SCHEMBL11537150 0.73 ALDH1A1 (0.42) ALDH1A1L3MBTL1CYP1A2CYP2C9CYP2C19
SCHEMBL11537148 0.73 ALDH1A1 (0.42) ALDH1A1L3MBTL1CYP1A2CYP2C9CYP2C19
SCHEMBL3850015 0.72 CES2 (0.56) ALDH1A1NPSR1PTGS2CES2CES1
SCHEMBL3850013 0.72 CES2 (0.56) ALDH1A1NPSR1PTGS2CES2CES1
SCHEMBL9155638 0.72 CES2 (0.61) ALDH1A1NPSR1PTGS2CES2CES1
SCHEMBL18885235 0.72 CES2 (0.55) ALDH1A1L3MBTL1CYP1A2CYP2C9CYP2C19
SCHEMBL9155633 0.72 CES2 (0.61) ALDH1A1NPSR1PTGS2CES2CES1
SCHEMBL8915867 0.71 ALDH1A1 (1.00) ALDH1A1L3MBTL1CYP1A2CYP2C9CYP2C19
SCHEMBL8689509 0.70 NPC1 (0.48) ALDH1A1PTGS2CES2CES1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0932600-A2 SULFONAMIDE SUBSTITUTED ASPARTIC ACID INTERLEUKIN-1$g(b) CONVERTING ENZYME INHIBITORS WARNER-LAMBERT COMPANY (US) 1999-08-04 EP disclosed
WO-1998016504-A2 SULFONAMIDE SUBSTITUTED ASPARTIC ACID INTERLEUKIN-1β CONVERTING ENZYME INHIBITORS WARNER-LAMBERT COMPANY (US) 1998-04-23 WO disclosed