SCHEMBL8562273

SCHEMBL8562273

COc1cccc(CN2CCC(Br)C2=O)c1

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.55
CMA1 P23946 1/20 0.54
KDM4E B2RXH2 3/20 0.52
ALDH1A1 P00352 3/20 0.52
MAPT P10636 2/20 0.51
PKM P14618 1/20 0.51
LMNA P02545 2/20 0.50
HTT P42858 1/20 0.50
KMT2A Q03164 1/20 0.50
ALOX15 P16050 1/20 0.49
TSHR P16473 1/20 0.49
OPRM1 P35372 1/20 0.48
ACHE P22303 1/20 0.47
GAA P10253 1/20 0.47
TP53 P04637 1/20 0.47
CES2 O00748 1/20 0.47
HRH3 Q9Y5N1 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8562278 1.00 SIGMAR1 (0.55) SIGMAR1CMA1KDM4EALDH1A1MAPT
SCHEMBL8562132 0.83 GAA (0.56) SIGMAR1CMA1ALDH1A1LMNAGAA
SCHEMBL8562128 0.83 GAA (0.56) SIGMAR1CMA1ALDH1A1LMNAGAA
SCHEMBL369615 0.83 ALDH1A1 (0.44) SIGMAR1CMA1KDM4EALDH1A1MAPT
SCHEMBL16885927 0.82 MEN1 (0.57) KDM4EALDH1A1HTTKMT2AACHE
SCHEMBL6828052 0.82 SIGMAR1 (0.56) SIGMAR1CMA1PKMKMT2A
SCHEMBL28961034 0.81 KMT2A (0.53) SIGMAR1CMA1KDM4EALDH1A1MAPT
SCHEMBL8567054 0.80 ALDH1A1 (0.55) SIGMAR1KDM4EALDH1A1KMT2AGAA
SCHEMBL8567056 0.80 ALDH1A1 (0.55) SIGMAR1KDM4EALDH1A1KMT2AGAA
SCHEMBL12494883 0.79 KMT2A (0.53) SIGMAR1CMA1KDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5804577-A ANTIBIOTICS HOFFMANN-LA ROCHE INC. (US) 1998-09-08 US disclosed
CN-1150950-A Cephalosporin derivatives HOFFMANN LA ROCHE (CH) 1997-06-04 CN disclosed
EP-0761673-A1 Cephalosporin derivatives F. HOFFMANN-LA ROCHE AG (CH) 1997-03-12 EP disclosed